10mM in DMSO for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Descripción general
ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1 / 2 inhibitor, showing 60% inhibition at 1 nM and an IC 50 of 3.0 nM against ERK1 and ERK2 , respectively
In Vitro
ERK1/2 inhibitor 1 (Compound 27) shows excellent antiproliferative potency with IC 50 s of 4.9 and 7.5 nM in A375 and Colo205 cells, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
IC50& Target:ERK2 3.0 nM (IC 50 ) ERK1
Specifications
Especificaciones y pureza
10mM in DMSO
Mecanismos bioquímicos y fisiológicos
ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1 / 2 inhibitor, showing 60% inhibition at 1 nM and an IC 50 of 3.0 nM against ERK1 and ERK2 , respectively.
Condiciones de almacenamiento de almacenamiento
Store at -80°C
Enviado en
Dry ice packs + Cold packs
Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.
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