BGC-20-1531 hydrochloride - ≥98% , CAS No.1962928-26-2

CAS: 1962928-26-2 Cat. No.: B288496 Molecular Weight: 529.00 PubChem CID: 121513858

GRADE & PURITY ≥98%

Synonyms

PGN 1531 | 4-[[4-(5-Methoxy-2-pyridinyl)phenoxy]methyl]-5-methyl-N-[(2-methylphenyl)sulfonyl]-2-furancarboxamide hydrochloride

Storage

Store at -20°C,Desiccated

Shipped In

Ice chest + Ice pads

Specifications

Synonyms

PGN 1531 | 4-[[4-(5-Methoxy-2-pyridinyl)phenoxy]methyl]-5-methyl-N-[(2-methylphenyl)sulfonyl]-2-furancarboxamide hydrochloride

Specifications & Purity

≥98%

Biochemical and Physiological Mechanisms

High affinity and selective EP4antagonist (Ki= 3 nM). Exhibits >2500-fold selectivity for EP4over EP2and EP3. Also selective over a range of other prostanoid receptors, ion channels, transporters and enzymes. Inhibits PGE2-induced vasodilation of middle c

Storage

Store at -20°C, Desiccated

Shipped In

Ice chest + Ice pads

This product requires cold chain shipping. Ground and other economy services are not available.

Action Type

ANTAGONIST

Purity

≥98%

Names and Identifiers

• Canonical Smiles: CC1=CC=CC=C1S(=O)(=O)NC(=O)C2=CC(=C(O2)C)COC3=CC=C(C=C3)C4=NC=C(C=C4)OC.Cl
• IUPAC Name: 4-[[4-(5-methoxypyridin-2-yl)phenoxy]methyl]-5-methyl-N-(2-methylphenyl)sulfonylfuran-2-carboxamide;hydrochloride
• InChIKey: ZSHYZCXOFPPBMH-UHFFFAOYSA-N
• INCHI: 1S/C26H24N2O6S.ClH/c1-17-6-4-5-7-25(17)35(30,31)28-26(29)24-14-20(18(2)34-24)16-33-21-10-8-19(9-11-21)23-13-12-22(32-3)15-27-23;/h4-15H,16H2,1-3H3,(H,28,29);1H
• Alternate CAS: 736183-35-0；1186532-61-5
• PubChem CID: 121513858
• Molecular Weight: 529.00

Chemical and Physical Properties

• Solubility: Solvent:DMSO, Max Conc. mg/mL: 49.25, Max Conc. mM: 100