Determine the necessary mass, volume, or concentration for preparing a solution.
| Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
|---|
224,000+ research products · Triple ISO certified · COA & SDS available for every product · Same-day shipping on in-stock items
Why this grade
Moligand™, ≥99% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
Storage & shipping
Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.
Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
Information
Tirzepatide (LY3298176) Tirzepatide (LY3298176, GIP/GLP-1 RA, TZP) is a dual GIP/GLP-1 receptor agonist. Tirzepatide differentially induces internalization of the GIP and GLP-1 receptors with EC50 values of 18.2 nM and 18.1 nM, respectively.
Specifications
Synonyms
GIP/GLP-1 RA | TZP
Specifications & Purity
Moligand™, ≥99%
Biochemical and Physiological Mechanisms
Tirzepatide (LY3298176, GIP/GLP-1 RA, TZP) is a dual GIP/GLP-1 receptor agonist. Tirzepatide differentially induces internalization of the GIP and GLP-1 receptors with EC50 values of 18.2 nM and 18.1 nM, respectively.
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Action Type
AGONIST
Mechanism of action
Agonist of GIP receptor;Agonist of GLP-1 receptor
Purity
≥99%
Names and Identifiers
| Molecular Weight | 4813.45(free) |
|---|
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
Download SDS →✅ Certificate of Analysis (COA)
Lot-specific quality data. Enter your lot number to retrieve the exact COA.
Look up COA →🔬 Specification Sheet
Full quality attributes and acceptance criteria for this grade.
View spec sheet →Advanced Data
Associated Targets(Human)
GIPR Tchem Gastric inhibitory polypeptide receptor (0 Activities)
GLP1R Tclin Glucagon-like peptide 1 receptor (0 Activities)
| Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
|---|
Certificates（CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Find and download the COA for your product by matching the lot number on the packaging.
| Lot Number | Certificate Type | Date | Item |
|---|---|---|---|
 F2603657 | Certificate of Analysis | May 22, 2026 | T412109 |
| F2603658 | Certificate of Analysis | May 22, 2026 | T412109 |
| F2603686 | Certificate of Analysis | May 22, 2026 | T412109 |
| F2603687 | Certificate of Analysis | May 22, 2026 | T412109 |
| F2603688 | Certificate of Analysis | May 22, 2026 | T412109 |
| G2417266 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417267 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417268 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417270 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417272 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417274 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417275 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417423 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417424 | Certificate of Analysis | Mar 29, 2024 | T412109 |
| G2417425 | Certificate of Analysis | Mar 29, 2024 | T412109 |
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Chemical and Physical Properties
| Solubility | Solubility (25°C) In vitro DMSO: 100 mg/mL (20.77 mM); Water: Insoluble; |
|---|
Solution Calculators
Reviews
Customer Reviews
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