GSK1521498 free base - 10mM in DMSO , CAS No.1007573-18-3

CAS: 1007573-18-3 Cat. No.: G655392 Molecular Weight: 402.44

GRADE & PURITY 10mM in DMSO

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Overview

GSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base has the potential for disorders of compulsive consumption of food, alcohol, and agents

IC50& Target:μ Opioid Receptor/MOR

Specifications

Specifications & Purity

10mM in DMSO

Biochemical and Physiological Mechanisms

GSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base has the potential for disorders of compulsive consumption of food, alcohol, and agents.

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

This product requires cold chain shipping. Ground and other economy services are not available.

Action Type

ANTAGONIST

Product Properties

• ALogP: 4.9

Names and Identifiers

• Isomeric SMILES: C1C(CC2=CC=CC=C21)NCC3=C(C=C(C=C3F)C4=CC(=CC=C4)C5=NC=NN5)F
• Alternate CAS: 1007573-18-3；1007578-24-6；1426543-84-1
• MeSH Entry Terms: GSK 1521498;GSK-1521498;GSK1521498;N-((3,5-difluoro-3'-(1H-1,2,4-triazol-3-yl)-4-biphenylyl)methyl)-2,3-dihydro-1H-inden-2-amine
• Molecular Weight: 402.44

Associated Targets(Human)

OPRM1 Tclin Mu-type opioid receptor (0 Activities)

Discover Target: OPRM1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)