S961 acetate - Moligand™,≥95% , CAS No.1083433-49-1(free basis)

CAS: 1083433-49-1(free basis) Cat. No.: S658830 Molecular Weight: 4802.12(free basis)

GRADE & PURITY Moligand™, ≥95%

Storage

Store at -20°C,Argon charged,Desiccated

Shipped In

Ice chest + Ice pads

Overview

S961 acetate is an high-affinity and selective insulin receptor ( IR ) antagonist with IC 50 s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively.

Appearance:Solid

In Vitro:S961 also shows high-affinity to Rat IR and Pig IR with IC 50 s of 0.056 nM and 0.084 nM in PEG-assay, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Biological Activity:S961 acetate is an high-affinity and selective insulin receptor ( IR ) antagonist with IC 50 s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively.

Specifications

Specifications & Purity

Moligand™, ≥95%

Storage

Store at -20°C, Argon charged, Desiccated

Shipped In

Ice chest + Ice pads

This product requires cold chain shipping. Ground and other economy services are not available.

Grade

Moligand™

Purity

≥95%

Names and Identifiers

• Molecular Weight: 4802.12(free basis)

Chemical and Physical Properties

• Solubility: DMSO : 12.5 mg/mL (2.57 mM; Need ultrasonic) H2O : 1.79 mg/mL (0.37 mM; ultrasonic and adjust pH to 8 with NaOH)
• Sensitivity: Moisture sensitive