CBP/p300-IN-10 - ≥98% , CAS No.2259641-71-7

CAS: 2259641-71-7 Cat. No.: C648970 Molecular Weight: 537.48
AVAILABLE TO ORDER
GRADE & PURITY ≥98%
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
 ·  off list, applied to all prices below.
Size
Status
Price
Qty
1mg
C648970-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$900.90
5mg
C648970-5mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$2,900.90
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Why this grade

≥98% for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Overview

CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC 50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer

In Vitro

CBP/p300-IN-10 (example 84) (0-1 μM; 3 h) inhibit H3K27Ac activity in LK2 cells with an IC 50 of 22 nM. CBP/p300-IN-10 (38 nM-10 mM; 3 days) has inhibitory activity against LK2 and TE-8. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Cell Proliferation AssayCell Line: LK2 and TE-8 Concentration: 38 nM-10 mM Incubation Time: 3 days Result: Inhibited LK2 and TE-8 with GI 50 s of 97.163 nM and 152.484 nM, respectively.

Form:Solid

IC50& Target:EP300 26 nM (IC 50 ) CREBBP 39 nM (IC 50 )

Specifications

Specifications & Purity
≥98%
Biochemical and Physiological Mechanisms
CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC 50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer.
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Action Type
INHIBITOR
Purity
≥98%
Names and Identifiers
Molecular Weight 537.48

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Certificates(CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
SolubilityDMSO : 10.5 mg/mL (19.54 mM; ultrasonic and warming and heat to 80°C)
Solution Calculators
Reviews

Customer Reviews

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