JMV1431, Antagonist of B 1 receptor;Antagonist of B 2 receptor, CAS No.284037-75-8, Antagonist of B 1 receptor;Antagonist of B 2 receptor

CAS: 284037-75-8 Cat. No.: rp174381 PubChem CID: 44316620

GRADE & PURITY Moligand™

Specifications

Product Name

JMV1431, Antagonist of B 1 receptor;Antagonist of B 2 receptor, CAS No.284037-75-8

Synonyms

JMV 1431;JMV-1431

Grade

Moligand™

Specifications & Purity

Moligand™

Action Type

ANTAGONIST

Mechanism of action

Antagonist of B 1 receptor;Antagonist of B 2 receptor

CAS

284037-75-8

Molecule Type

Small molecule

Storage and Shipping

Storage

Room temperature

Taxonomic Classification

Taxonomy Tree

• Kingdom Organic compounds
  • Superclass Organic acids and derivatives
    • Class Carboxylic acids and derivatives
      • Subclass Amino acids, peptides, and analogues
        • Level5 Peptides
          • Level6 Oligopeptides

• Kingdom: Organic compounds
• Superclass: Organic acids and derivatives
• Class: Carboxylic acids and derivatives
• Subclass: Amino acids, peptides, and analogues
• Intermediate Tree Nodes: Peptides
• Direct Parent: Oligopeptides
• Alternative Parents: N-acyl-alpha amino acids and derivatives Proline and derivatives Serine and derivatives Alpha amino acid amides Benzothiazepines N-acylpyrrolidines Pyrrolidinecarboxamides Alkylarylthioethers Benzenoids N-acyl amines Tertiary carboxylic acid amides Heteroaromatic compounds Thiophenes Secondary carboxylic acid amides Guanidines Lactams Amino acids Secondary alcohols Propargyl-type 1,3-dipolar organic compounds Azacyclic compounds Monocarboxylic acids and derivatives Carboximidamides Carboxylic acids Monoalkylamines Carbonyl compounds Primary alcohols Organic oxides Hydrocarbon derivatives
• Molecular Framework: Aromatic heteropolycyclic compounds
• Substituents: Alpha-oligopeptide - N-acyl-alpha amino acid or derivatives - Proline or derivatives - Alpha-amino acid amide - Serine or derivatives - Benzothiazepine - N-substituted-alpha-amino acid - Alpha-amino acid or derivatives - Pyrrolidine-2-carboxamide - Pyrrolidine carboxylic acid or derivatives - N-acylpyrrolidine - Aryl thioether - Alkylarylthioether - Benzenoid - Fatty acyl - N-acyl-amine - Fatty amide - Tertiary carboxylic acid amide - Thiophene - Pyrrolidine - Heteroaromatic compound - Amino acid or derivatives - Amino acid - Carboxamide group - Guanidine - Lactam - Secondary alcohol - Secondary carboxylic acid amide - Thioether - Carboximidamide - Propargyl-type 1,3-dipolar organic compound - Carboxylic acid - Monocarboxylic acid or derivatives - Azacycle - Organoheterocyclic compound - Organic 1,3-dipolar compound - Organic oxide - Hydrocarbon derivative - Alcohol - Organic oxygen compound - Carbonyl group - Amine - Primary aliphatic amine - Primary amine - Primary alcohol - Organic nitrogen compound - Organonitrogen compound - Organooxygen compound - Aromatic heteropolycyclic compound
• Description: This compound belongs to the class of organic compounds known as oligopeptides. These are organic compounds containing a sequence of between three and ten alpha-amino acids joined by peptide bonds.
• External Descriptors: Not available

Data sources

1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.

DOI: 10.1186/s13321-016-0174-y

Associated Targets(Human)

BDKRB2 Tclin B2 bradykinin receptor (1 Activities)

Discover Target: BDKRB2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

BDKRB1 Tchem B1 bradykinin receptor (1 Activities)

Discover Target: BDKRB1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

BDKRB2 Tclin Bradykinin B2 receptor (3970 Activities)

Discover Target: BDKRB2

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Bdkrb1 Bradykinin B1 receptor (77 Activities)

Discover Target: Bdkrb1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Genetic information

• Alternate Names: JMV 1431;JMV-1431
• Reference:
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