PRL-2915, Antagonist of SST 2 receptor;Antagonist of SST 3 receptor;Antagonist of SST 4 receptor;Antagonist of SST 5 receptor, CAS No.209006-18-8, Antagonist of SST 2 receptor;Antagonist of SST 3 receptor;Antagonist of SST 4 receptor;Antagonist of SST 5 receptor

CAS: 209006-18-8 Cat. No.: rp174803 PubChem CID: 10677800

GRADE & PURITY Moligand™

Specifications

Product Name

PRL-2915, Antagonist of SST 2 receptor;Antagonist of SST 3 receptor;Antagonist of SST 4 receptor;Antagonist of SST 5 receptor, CAS No.209006-18-8

Synonyms

PRL 2915

Grade

Moligand™

Specifications & Purity

Moligand™

Action Type

ANTAGONIST

Mechanism of action

Antagonist of SST 2 receptor;Antagonist of SST 3 receptor;Antagonist of SST 4 receptor;Antagonist of SST 5 receptor

CAS

209006-18-8

Molecule Type

Peptide

Storage and Shipping

Storage

Room temperature

Taxonomic Classification

Taxonomy Tree

• Kingdom Organic compounds
  • Superclass Organic acids and derivatives
    • Class Carboxylic acids and derivatives
      • Subclass Amino acids, peptides, and analogues
        • Level5 Peptides
          • Level6 Oligopeptides

• Kingdom: Organic compounds
• Superclass: Organic acids and derivatives
• Class: Carboxylic acids and derivatives
• Subclass: Amino acids, peptides, and analogues
• Intermediate Tree Nodes: Peptides
• Direct Parent: Oligopeptides
• Alternative Parents: Cyclic peptides Phenylalanine and derivatives Macrolactams N-acyl-alpha amino acids and derivatives Alpha amino acid amides 3-alkylindoles Naphthalenes Amphetamines and derivatives Aralkylamines Chlorobenzenes Aryl chlorides Fatty amides Substituted pyrroles Pyridines and derivatives Heteroaromatic compounds Secondary carboxylic acid amides Organic disulfides Lactams Primary carboxylic acid amides Azacyclic compounds Carbonyl compounds Hydrocarbon derivatives Monoalkylamines Organic oxides Organochlorides
• Molecular Framework: Aromatic heteropolycyclic compounds
• Substituents: Alpha-oligopeptide - Cyclic alpha peptide - Phenylalanine or derivatives - N-acyl-alpha amino acid or derivatives - Macrolactam - Alpha-amino acid amide - N-substituted-alpha-amino acid - Alpha-amino acid or derivatives - Amphetamine or derivatives - Naphthalene - 3-alkylindole - Indole or derivatives - Indole - Aralkylamine - Halobenzene - Chlorobenzene - Aryl chloride - Fatty acyl - Pyridine - Monocyclic benzene moiety - Fatty amide - Substituted pyrrole - Benzenoid - Aryl halide - Pyrrole - Heteroaromatic compound - Amino acid or derivatives - Secondary carboxylic acid amide - Carboxamide group - Primary carboxylic acid amide - Lactam - Organic disulfide - Organoheterocyclic compound - Azacycle - Organooxygen compound - Primary amine - Amine - Organic oxide - Carbonyl group - Organic oxygen compound - Organonitrogen compound - Organochloride - Organohalogen compound - Organic nitrogen compound - Hydrocarbon derivative - Primary aliphatic amine - Aromatic heteropolycyclic compound
• Description: This compound belongs to the class of organic compounds known as oligopeptides. These are organic compounds containing a sequence of between three and ten alpha-amino acids joined by peptide bonds.
• External Descriptors: Not available

Data sources

1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.

DOI: 10.1186/s13321-016-0174-y

Associated Targets(Human)

SSTR2 Tclin Somatostatin receptor type 2 (0 Activities)

Discover Target: SSTR2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

SSTR3 Tclin Somatostatin receptor type 3 (0 Activities)

Discover Target: SSTR3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

SSTR4 Tclin Somatostatin receptor type 4 (0 Activities)

Discover Target: SSTR4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

SSTR5 Tclin Somatostatin receptor type 5 (0 Activities)

Discover Target: SSTR5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Genetic information

• Alternate Names: PRL 2915
• Reference:
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  • 30. Integrative predictive model of coronary artery calcification in atherosclerosis., Circulation, McGeachie, Michael M and 13 more authors.
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  • 76. Augmented H2S production via cystathionine-beta-synthase upregulation plays a role in pregnancy-associated uterine vasodilation., Biology of reproduction, Sheibani, Lili L and 7 more authors.
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