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GSK256073 - Moligand™,≥99% , CAS No.862892-90-8

CAS: 862892-90-8 Cat. No.: G646139 Molecular Weight: 256.69 EC Number: 629-897-2 PubChem CID: 46215799
COA
GSK256073 - ≥99% CAS No(862892-90-8) by Aladdin Scientific
AVAILABLE TO ORDER
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥99%
Synonyms
GTPL8470 | E80530 | GSK 256073 | SCHEMBL2473169 | 862892-90-8 (free) | DTXSID80673110 | OKL | 1571098-00-4 | 1H-Purine-2,6-dione, 8-chloro-3,9-dihydro-3-pentyl- | 8-chloro-3-pentyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione | A931950 | 8-chloranyl-3-pentyl-7H
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
★
 ·  off list, applied to all prices below.
Size
Status
Price
Qty
5mg
G646139-5mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$146.90
1mg
G646139-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$59.90
10mg
G646139-10mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$236.90
25mg
G646139-25mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$416.90
50mg
G646139-50mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$612.90
100mg
G646139-100mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$869.90
1g
G646139-1g
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$239.90
5g
G646139-5g
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$839.90
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SDS
Safety data
COA
Certificate
DS
Datasheet
SP
Spec sheet
Specifications Names and Identifiers Documentation Advanced Data Taxonomic Classification 3D Structure Associated Targets(Human) Mechanisms of Action Certificates（CoA,COO,BSE/TSE and Analysis Chart) Chemical and Physical Properties Solution Calculators Reviews
🧪

Why this grade

Moligand™,≥99% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

🌡

Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

📚

Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Specifications

Synonyms
GTPL8470 | E80530 | GSK 256073 | SCHEMBL2473169 | 862892-90-8 (free) | DTXSID80673110 | OKL | 1571098-00-4 | 1H-Purine-2, 6-dione, 8-chloro-3, 9-dihydro-3-pentyl- | 8-chloro-3-pentyl-2, 3, 6, 7-tetrahydro-1H-purine-2, 6-dione | A931950 | 8-chloranyl-3-pentyl-7H
Specifications & Purity
Moligand™, ≥99%
Biochemical and Physiological Mechanisms
GSK26073 is a potent and selective GPR109A agonist, as well as a long-acting, non flushing HCA2 complete agonist with a pEC 50 of 7.5 (human HCA2). GSK256073 can improve glucose homeostasis by inhibiting fat decomposition, and may be used to treat diabete
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Action Type
AGONIST
Purity
≥99%
Names and Identifiers
Canonical SmilesCCCCCN1C2=C(C(=O)NC1=O)NC(=N2)Cl
IUPAC Name8-chloro-3-pentyl-7H-purine-2,6-dione
InChIKeyCGAMDQCXAAOFSR-UHFFFAOYSA-N
INCHI1S/C10H13ClN4O2/c1-2-3-4-5-15-7-6(12-9(11)13-7)8(16)14-10(15)17/h2-5H2,1H3,(H,12,13)(H,14,16,17)
Isomeric SMILES CCCCCN1C2=C(C(=O)NC1=O)NC(=N2)Cl
Alternate CAS 862892-90-8
PubChem CID 46215799
MeSH Entry Terms 8-chloro-3-pentyl-1H-purine-2,6(3H,7H)-dione;GSK256073
Molecular Weight 256.69

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

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🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

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Advanced Data

Taxonomic Classification

Taxonomy Tree

KingdomOrganic compounds
SuperclassOrganoheterocyclic compounds
ClassImidazopyrimidines
SubclassPurines and purine derivatives
Intermediate Tree Nodes Not available
Direct ParentXanthines
Alternative Parents 6-oxopurines  Alkaloids and derivatives  Pyrimidones  Aryl chlorides  Vinylogous amides  Imidazoles  Heteroaromatic compounds  Ureas  Lactams  Azacyclic compounds  Organooxygen compounds  Organonitrogen compounds  Organochlorides  Organic oxides  Hydrocarbon derivatives  
Molecular FrameworkAromatic heteropolycyclic compounds
Substituents Xanthine - 6-oxopurine - Purinone - Alkaloid or derivatives - Pyrimidone - Aryl chloride - Aryl halide - Pyrimidine - Azole - Heteroaromatic compound - Imidazole - Vinylogous amide - Lactam - Urea - Azacycle - Organonitrogen compound - Organochloride - Organohalogen compound - Organic nitrogen compound - Hydrocarbon derivative - Organic oxide - Organic oxygen compound - Organooxygen compound - Aromatic heteropolycyclic compound
DescriptionThis compound belongs to the class of organic compounds known as xanthines. These are purine derivatives with a ketone group conjugated at carbons 2 and 6 of the purine moiety.
External Descriptors Not available
3D Structure
Interactive Chemical Structure Model





Associated Targets(Human)
HCAR2 Tclin Hydroxycarboxylic acid receptor 2 (0 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
Mechanisms of Action
Certificates（CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
SolubilityDMSO : 16.67 mg/mL (64.94 mM; Need ultrasonic)
Molecular Weight256.690 g/mol
XLogP32.300
Hydrogen Bond Donor Count2
Hydrogen Bond Acceptor Count3
Rotatable Bond Count4
Exact Mass256.073 Da
Monoisotopic Mass256.073 Da
Topological Polar Surface Area78.100 Ų
Heavy Atom Count17
Formal Charge0
Complexity325.000
Isotope Atom Count0
Defined Atom Stereocenter Count0
Undefined Atom Stereocenter Count0
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
The total count of all stereochemical bonds0
Covalently-Bonded Unit Count1
Solution Calculators
Reviews

Customer Reviews

Need help choosing the grade?

Our grade selection guide covers purity, stabilizer status, and application suitability for all variants in our catalog.

View Moligand™ grade guide →
Bulk & Custom Packaging Need larger quantities or custom specifications? Contact our team for a tailored quote.

View related series

Class A GPCR (8120) GPCR/G Protein (3180) GPR109A (7)

Related Products

GSK256073 - Moligand™,10mM in DMSO , CAS No.862892-90-8
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