PROTAC BRD4-binding moiety 1 , CAS No.2101200-10-4

CAS: 2101200-10-4 Cat. No.: P651455 Molecular Weight: 371.43 PubChem CID: 141488040
AVAILABLE TO ORDER
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
 ·  off list, applied to all prices below.
Size
Status
Price
Qty
10mg
P651455-10mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$1,314.90
25mg
P651455-25mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$2,630.90
5mg
P651455-5mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$820.90
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Why this grade

for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

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Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Overview

PROTAC BRD4-binding moiety 1 is a ligand for BRD4 . PROTAC BRD4-binding moiety 1 binds to cereblon ligand via a linker to form PROTAC to degrade BRD4

In Vitro

PROTAC BRD4 Degrader-2 is an efficacious PROTAC BRD4 degrader with an IC 50 of 14.2 nM against BRD4 BD1. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:BRD4

Specifications

Biochemical and Physiological Mechanisms
PROTAC BRD4-binding moiety 1 is a ligand for BRD4 . PROTAC BRD4-binding moiety 1 binds to cereblon ligand via a linker to form PROTAC to degrade BRD4 ( HY-133136 ).
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Names and Identifiers
Isomeric SMILES CC1=C(C(=NO1)C)C2=CC3=C(C=C2)N(C(=O)N(C3C4=CC=CC=C4)CC#C)C
PubChem CID 141488040
Molecular Weight 371.43

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Certificates(CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Solution Calculators
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