Sar-[D-Phe8]-des-Arg9-Bradykinin TFA salt, Agonist of B 1 receptor, CAS No.126959-88-4(free base), Agonist of B 1 receptor

CAS: 126959-88-4(free base) Cat. No.: S287120 Molecular Weight: 975.11(free base)

GRADE & PURITY Moligand™, ≥98%

Specifications

Product Name

Sar-[D-Phe8]-des-Arg9-Bradykinin TFA salt, Agonist of B 1 receptor, CAS No.126959-88-4(free base)

Grade

Moligand™

Specifications & Purity

Moligand™, ≥98%

Biochemical and Physiological Mechanisms

Potent and selective bradykinin B1receptor agonist (EC50= 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cleavage. Exhibits hypotensive and angiogenic activityin vivo.

Sequence

XRPPGFSPF(Modifications: X = Sar, Phe-9 = D-Phe)

Action Type

AGONIST

Mechanism of action

Agonist of B 1 receptor

CAS

126959-88-4(free base)

Molecule Type

Peptide

Storage and Shipping

Storage

Store at -20°C,Desiccated

Shipped In

Ice chest + Ice pads

Associated Targets(Human)

BDKRB1 Tchem B1 bradykinin receptor (0 Activities)

Discover Target: BDKRB1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Genetic information

• Reference:
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