≥98% for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at 2-8°C,Protected from light Ships Wet ice Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
4,5-Dimethoxycanthin-6-one is a potent and uncompetitive inhibitor of CYP1A2 -mediated phenacetin O-deethylation with an IC 50 value of 1.7μM and a K i value of 2.6 μM. 4,5-Dimethoxycanthin-6-one, as an alkaloid, is isolated from the wood of Picrasma quassioides BENNET (Simaroubaceae).
In Vitro
4,5-Dimethoxycanthin-6-one is a potent and uncompetitive inhibitor of CYP1A2-mediated phenacetin O-deethylation with an IC 50 value of 1.7μM and a K i value of 2.6 μM. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Form:Solid
Specifications
Specifications & Purity
≥98%
Biochemical and Physiological Mechanisms
4, 5-Dimethoxycanthin-6-one is a potent and uncompetitive inhibitor of CYP1A2 -mediated phenacetin O-deethylation with an IC 50 value of 1.7μM and a K i value of 2.6 μM. 4, 5-Dimethoxycanthin-6-one, as an alkaloid, is isolated from the wood of Picrasma quas
Storage
Store at 2-8°C, Protected from light
Shipped In
Wet ice
This product requires cold chain shipping. Ground and other economy services are not available.
Action Type
INHIBITOR
Purity
≥98%
Names and Identifiers
Isomeric SMILES
COC1=C(C(=O)N2C3=CC=CC=C3C4=C2C1=NC=C4)OC
PubChem CID
638215
Molecular Weight
280.28
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
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