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CB1/2 agonist 3 - ≥99% , CAS No.2772655-86-2
AVAILABLE TO ORDER
GRADE & PURITY ≥99%
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
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Why this grade
≥99% for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
Storage & shipping
Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.
Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
CB1/2 agonist 3 (compound 52), a potent non-selective cannabinoid ligand, is a CB1/CB2 (cannabinoid receptor) competitive agonist. CB1/2 agonist 3 acts on hCB1 and hCB2 with K i values of 5.9 nM and 3.5 nM, respectively .
Form:Solid
IC50& Target:hCB1-R 5.9 nM (Ki) hCB2-R 3.5 nM (Ki)
In Vitro:CB1/2 agonist 3 (compound 52) can partially induce [ 35 S]GTPγS binding to hCB1-CHO cell membranes with an EC 50 value of 30.99 nM, and slightly inhibit [ 35 S]GTPγS binding to hCB2-CHO cell membranes with a mean EC 50 value of 1.28 nM . CB1/2 agonist 3 (compound 52) ((1 μM, 1 h) has antagonistic effect on CB1/CB2 agonist CP-55940 with a K b value of 78.17 nM. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Specifications
Specifications & Purity
≥99%
Biochemical and Physiological Mechanisms
CB1/2 agonist 3 (compound 52), a potent non-selective cannabinoid ligand, is a CB1/CB2 (cannabinoid receptor) competitive agonist. CB1/2 agonist 3 acts on hCB1 and hCB2 with K i values of 5.9 nM and 3.5 nM, respectively.
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Action Type
AGONIST
Purity
≥99%
Names and Identifiers
| Molecular Weight | 387.60 |
|---|
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
Download SDS →✅ Certificate of Analysis (COA)
Lot-specific quality data. Enter your lot number to retrieve the exact COA.
Look up COA →🔬 Specification Sheet
Full quality attributes and acceptance criteria for this grade.
View spec sheet →Advanced Data
Certificates（CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
| Solubility | DMSO : 10 mg/mL (25.80 mM; Need ultrasonic) |
|---|
Solution Calculators
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