10mM in DMSO for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
Clopidogrel thiolactone is an active metabolites containing thiols resulting from thionolactone transformation of clopidogrel . Clopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent
In Vivo
Clopidogrel thiolactone (8 μm/kg; i.v.; Sprague-Dawley male rats) has good biological availability and pharmacokinetic parameters . MCE has not independently confirmed the accuracy of these methods. They are for reference only. Animal Model: Sprague-Dawley male rats Dosage: 8 μm/kg; orally clopidogrel (24 μm/kg) Administration: Intravenous injection; collected blood at 0 h (before dosing) and 0.083, 0.167, 0.5, 1, 2, 4, 6, 8, 24 h postdose. Result: 1.19 Parameter Clopidogrel C max (μg/L) 6.93 T max (h) 0.583 t 1/2 (h) 2.48 AUC 0-∞ (μg*h/L) 32.2
IC50& Target:P2Y12 Receptor
Specifications
Specifications & Purity
10mM in DMSO
Biochemical and Physiological Mechanisms
Clopidogrel thiolactone is an active metabolites containing thiols resulting from thionolactone transformation of clopidogrel ( HY-15283 ). Clopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent.
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
This product requires cold chain shipping. Ground and other economy services are not available.
Action Type
INHIBITOR
Names and Identifiers
Isomeric SMILES
COC(=O)[C@H](C1=CC=CC=C1Cl)N2CCC3C(=CC(=O)S3)C2
PubChem CID
56848893
Molecular Weight
337.82
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
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