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LPA2 antagonist 1 - Moligand™,10mM in DMSO , CAS No.1017606-66-4

CAS: 1017606-66-4 Cat. No.: L656453 Molecular Weight: 500.46
COA
LPA2 antagonist 1 - 10mM in DMSO CAS No(1017606-66-4) by Aladdin Scientific
AVAILABLE TO ORDER
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. 10mM in DMSO
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
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 ·  off list, applied to all prices below.
Size
Status
Price
Qty
1ml
L656453-1ml
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$289.90
1mg
L656453-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$109.90
25mg
L656453-25mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$749.90
100mg
L656453-100mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$1,469.90
250mg
L656453-250mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$2,569.90
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SDS
Safety data
COA
Certificate
DS
Datasheet
SP
Spec sheet
Overview Specifications Names and Identifiers Documentation Advanced Data Associated Targets(Human) Certificates（CoA,COO,BSE/TSE and Analysis Chart) Solution Calculators Reviews
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Why this grade

Moligand™,10mM in DMSO Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

🌡

Storage & shipping

Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

📚

Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Overview

LPA2 antagonist 1 is a LPA2 antagonist with an IC 50 of 17 nM.

In Vitro

LPA2 antagonist 1 inhibits the phosphorylation of Erk induced by LPA in a concentration dependent manner. LPA2 antagonist 1 inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

IC50& Target:IC50: 17 nM (LPA2)

Specifications

Specifications & Purity
Moligand™, 10mM in DMSO
Biochemical and Physiological Mechanisms
LPA2 antagonist 1 is a LPA2 antagonist with an IC 50 of 17 nM.
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Action Type
INHIBITOR
Names and Identifiers
Isomeric SMILES CC1=CSC2=C1N=CN=C2N[C@@H](C)CN3CCN(CC3)S(=O)(=O)C4=CC(=C(C=C4)Cl)Cl
Molecular Weight 500.46

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Associated Targets(Human)
LPAR2 Tchem Lysophosphatidic acid receptor 2 (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
Certificates（CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Solution Calculators
Reviews

Customer Reviews

Need help choosing the grade?

Our grade selection guide covers purity, stabilizer status, and application suitability for all variants in our catalog.

View Moligand™ grade guide →
Bulk & Custom Packaging Need larger quantities or custom specifications? Contact our team for a tailored quote.

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