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224,000+ research products · Triple ISO certified · COA & SDS available for every product · Same-day shipping on in-stock items MBX-2982 - Moligand™, ≥98% , Glucose-dependent insulinotropic receptor agonist, CAS No.1037792-44-1, Glucose-dependent insulinotropic receptor agonist
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98% Synonyms
MBX 2982 | EX-A1003 | MBX2982 | MBX-2982 | DTXSID20146055 | AMY39989 | BDBM50013909 | MFCD22628771 | 8VP | 2-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-4-[[4-(1,2,3,4-tetrazol-1-yl)phenoxy]methyl]-1,3-thiazole | B5TRY67L51 | 4-((4-(1H-tetrazol-1-yl)phenoxy
Shipped In
Ice chest + Ice pads
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Why this grade Moligand™, ≥98% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.
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Quality documents SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview MBX-2982 is a selective, orally-available GPR119 agonist for the treatment of type 2 tiabetes.
Specifications Synonyms
MBX 2982 | EX-A1003 | MBX2982 | MBX-2982 | DTXSID20146055 | AMY39989 | BDBM50013909 | MFCD22628771 | 8VP | 2-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-4-[[4-(1, 2, 3, 4-tetrazol-1-yl)phenoxy]methyl]-1, 3-thiazole | B5TRY67L51 | 4-((4-(1H-tetrazol-1-yl)phenoxy
Specifications & Purity
Moligand™, ≥98%
Biochemical and Physiological Mechanisms
MBX-2982 is a potential first-in-class treatment for type 2 diabetes that targets G protein-coupled receptor 119 (GPR119), a receptor that interacts with bioactive lipids known to stimulate glucose-dependent insulin secretion. Preclinical data indicate th
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Mechanism of action
Glucose-dependent insulinotropic receptor agonist
Product Properties Names and Identifiers Canonical Smiles CCC1=CN=C(N=C1)N2CCC(CC2)C3=NC(=CS3)COC4=CC=C(C=C4)N5C=NN=N5 IUPAC Name 2-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-4-[[4-(tetrazol-1-yl)phenoxy]methyl]-1,3-thiazole InChIKey NFTMKHWBOINJGM-UHFFFAOYSA-N INCHI 1S/C22H24N8OS/c1-2-16-11-23-22(24-12-16)29-9-7-17(8-10-29)21-26-18(14-32-21)13-31-20-5-3-19(4-6-20)30-15-25-27-28-30/h3-6,11-12,14-15,17H,2,7-10,13H2,1H3 Isomeric SMILES CCC1=CN=C(N=C1)N2CCC(CC2)C3=NC(=CS3)COC4=CC=C(C=C4)N5C=NN=N5 Molecular Weight 448.54 Reaxy-Rn 18425804 Reaxys-RN_link_address https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=18425804&ln=
Documentation 📋 Safety Data Sheet (SDS) Comprehensive hazard, handling, storage, and regulatory compliance document.
Download SDS → ✅ Certificate of Analysis (COA) Lot-specific quality data. Enter your lot number to retrieve the exact COA.
Look up COA → 📊 Datasheet Quick-reference summary of product specifications and applications.
View datasheet → 🔬 Specification Sheet Full quality attributes and acceptance criteria for this grade.
View spec sheet →
Advanced Data Taxonomic Classification Kingdom Organic compounds Superclass Organoheterocyclic compounds Class Azoles Subclass Tetrazoles Intermediate Tree Nodes Not available Direct Parent Phenyltetrazoles and derivatives Alternative Parents Phenoxy compounds Phenol ethers Dialkylarylamines Aminopyrimidines and derivatives Alkyl aryl ethers 2,4-disubstituted thiazoles Piperidines Heteroaromatic compounds Azacyclic compounds Hydrocarbon derivatives Molecular Framework Aromatic heteromonocyclic compounds Substituents Phenyltetrazole - Phenoxy compound - Phenol ether - Dialkylarylamine - 2,4-disubstituted 1,3-thiazole - Alkyl aryl ether - Aminopyrimidine - Monocyclic benzene moiety - Piperidine - Pyrimidine - Benzenoid - Heteroaromatic compound - Thiazole - Azacycle - Ether - Organooxygen compound - Organonitrogen compound - Organic nitrogen compound - Organic oxygen compound - Amine - Hydrocarbon derivative - Aromatic heteromonocyclic compound Description This compound belongs to the class of organic compounds known as phenyltetrazoles and derivatives. These are compounds containing a phenyltetrazole skeleton, which consists of a tetrazole bound to a phenyl group. External Descriptors Not available Data sources 1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.
3D Structure Associated Targets(Human) Associated Targets(non-human) Mechanisms of Action Certificates(CoA,COO,BSE/TSE and Analysis Chart) Chemical and Physical Properties Solubility DMSO Molecular Weight 448.500 g/mol XLogP3 3.600 Hydrogen Bond Donor Count 0 Hydrogen Bond Acceptor Count 9 Rotatable Bond Count 7 Exact Mass 448.179 Da Monoisotopic Mass 448.179 Da Topological Polar Surface Area 123.000 Ų Heavy Atom Count 32 Formal Charge 0 Complexity 564.000 Isotope Atom Count 0 Defined Atom Stereocenter Count 0 Undefined Atom Stereocenter Count 0 Defined Bond Stereocenter Count 0 Undefined Bond Stereocenter Count 0 The total count of all stereochemical bonds 0 Covalently-Bonded Unit Count 1
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