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RX-3117 - Moligand™, ≥98% , CAS No.865838-26-2
AVAILABLE TO ORDER
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Why this grade
Moligand™, ≥98% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
Storage & shipping
Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.
Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
RX-3117 (fluorocyclopentenylcytosine) is a novel a cytidine analog. RX-3117 displays anticancer activity in several cancer cell lines, including gemcitabine-resistant variants.
Specifications
Synonyms
TV-1360 | Fluorocyclopentenylcytosine
Specifications & Purity
Moligand™, ≥98%
Biochemical and Physiological Mechanisms
RX-3117 (TV-1360) is a potent and active anti-cancer and anti metabolic agent. RX-3117 can inhibit DNA methyltransferase 1 (DNMT1). RX-3117 has anti proliferative and anti-tumor activities. RX-3117 can induce cell cycle arrest in the S phase and lead to c
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Action Type
INHIBITOR
Purity
≥98%
Names and Identifiers
| Isomeric SMILES | C1=CN(C(=O)N=C1N)[C@H]2[C@@H]([C@@H](C(=C2F)CO)O)O |
|---|---|
| PubChem CID | 11242315 |
| Molecular Weight | 257.22 |
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
Download SDS →✅ Certificate of Analysis (COA)
Lot-specific quality data. Enter your lot number to retrieve the exact COA.
Look up COA →🔬 Specification Sheet
Full quality attributes and acceptance criteria for this grade.
View spec sheet →Advanced Data
Associated Targets(Human)
HT-29 (80576 Activities)
K562 (73714 Activities)
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MCF7 (126967 Activities)
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MKN-45 (2102 Activities)
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OVCAR-3 (48710 Activities)
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PANC-1 (6144 Activities)
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PC-3 (62116 Activities)
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SK-MEL-28 (48833 Activities)
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U-251 (51189 Activities)
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A549 (127892 Activities)
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HCT-116 (91556 Activities)
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HepG2 (196354 Activities)
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LNCaP (8286 Activities)
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HeLa (62764 Activities)
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MDA-MB-231 (73002 Activities)
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NCI-H226 (44470 Activities)
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Associated Targets(non-human)
Hdac6 Histone deacetylase 6 (222 Activities)
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Mus musculus (284745 Activities)
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rep Replicase polyprotein 1ab (378 Activities)
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Mechanisms of Action
Certificates（CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
| Solubility | DMSO : ≥ 50 mg/mL (194.39 mM) |
|---|---|
| Molecular Weight | 257.220 g/mol |
| XLogP3 | -2.600 |
| Hydrogen Bond Donor Count | 4 |
| Hydrogen Bond Acceptor Count | 5 |
| Rotatable Bond Count | 2 |
| Exact Mass | 257.081 Da |
| Monoisotopic Mass | 257.081 Da |
| Topological Polar Surface Area | 119.000 Ų |
| Heavy Atom Count | 18 |
| Formal Charge | 0 |
| Complexity | 474.000 |
| Isotope Atom Count | 0 |
| Defined Atom Stereocenter Count | 3 |
| Undefined Atom Stereocenter Count | 0 |
| Defined Bond Stereocenter Count | 0 |
| Undefined Bond Stereocenter Count | 0 |
| The total count of all stereochemical bonds | 0 |
| Covalently-Bonded Unit Count | 1 |
Solution Calculators
Reviews
Customer Reviews
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