10mM in DMSO for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
SGK1-IN-1 is a highly active and selective inhibitor of SGK-1 , with an IC 50 of 1 nM.
In Vitro
SGK1-IN-1 (14n) shows an acceptable SGK isoform selectivity with a good activity on hSGK2 and a moderate activity on the hSGK3, with IC 50 s of 1, 41 nM at 10 μM and 50 μM ATP concentration, respectively. SGK1-IN-1 also displays cellular activity in a SGK1-dependent phosphorylation of GSK3β assay in U2OS cells with activities of 0.69 μM. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
IC50& Target:SGK1
Specifications
Specifications & Purity
10mM in DMSO
Biochemical and Physiological Mechanisms
SGK1-IN-1 is a highly active and selective inhibitor of SGK-1 , with an IC 50 of 1 nM.
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
This product requires cold chain shipping. Ground and other economy services are not available.
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