[Met5]-Enkephalin, amide TFA - ≥98% , CAS No.60117-17-1(free base)

CAS: 60117-17-1(free base) Cat. No.: M274977 Molecular Weight: 572.69(free base)

GRADE & PURITY ≥98%

Synonyms

HY-P1467 | Enkephalinamide-met- | (2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanamide | H-Tyr-Gly-Gly-Phe-Met-NH2 | 14-Amino-5-benzyl-4,7,10,13-tetrahydro

Storage

Protected from light,Store at -20°C

Shipped In

Ice chest + Ice pads

Overview

[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) (60117-17-1 free base) is a delta opioid receptor agonist and a presumed zeta opioid receptor.

Specifications

Synonyms

HY-P1467 | Enkephalinamide-met- | (2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanamide | H-Tyr-Gly-Gly-Phe-Met-NH2 | 14-Amino-5-benzyl-4, 7, 10, 13-tetrahydro

Specifications & Purity

≥98%

Biochemical and Physiological Mechanisms

Opioid peptide, with agonist activity at μ and δ receptors. Growth factor. Competes and mimics effects of opiate drugs. Stimulates intestinal ion transport. Neurotransmitter and neuromodulator. Active in vivo and in vitro .

Storage

Protected from light, Store at -20°C

Shipped In

Ice chest + Ice pads

This product requires cold chain shipping. Ground and other economy services are not available.

Note

Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one week. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

Purity

≥98%

Names and Identifiers

• Alternate CAS: 2918768-28-0
• Molecular Weight: 572.69(free base)
• Reaxy-Rn: 4284576
• Reaxys-RN_link_address: https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=4284576&ln=

Associated Targets(Human)

OPRM1 Tclin Mu opioid receptor (19785 Activities)

Discover Target: OPRM1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

OPRD1 Tclin Delta opioid receptor (15096 Activities)

Discover Target: OPRD1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

OPRK1 Tclin Kappa opioid receptor (16155 Activities)

Discover Target: OPRK1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Chemical and Physical Properties

• Solubility: Soluble in water
• Sensitivity: Moisture sensitiv；Light sensitive