Erastin - Moligand™, ≥99% , CAS No.571203-78-6

CAS: 571203-78-6 Cat. No.: E126853 Peso molecular: 547.04 Número EC: 637-217-0
Disponible para pedir
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥99%
Synonyms
2-(1-(4-(2-(4-chlorophenoxy)acetyl)piperazin-1-yl)ethyl)-3-(2-ethoxyphenyl)quinazolin-4(3H)-one | MFCD09837984 | 2-[1-[4-[2-(4-chlorophenoxy)acetyl]-1-piperazinyl]ethyl]-3-(2-ethoxyphenyl)-4(3H)-Quinazolinone | 2-(1-(4-(2-(4-Chlorophenoxy)acetyl)-1-pipera
Storage
Store at -20°C,Argon charged
Shipped In
Ice chest + Ice pads
 ·  off list, applied to all prices below.
Size
Estado
Price
Qty
5mg
E126853-5mg
3

33,90US$

50,90US$
Guardar 17,00 US$ (33.40%)
25mg
E126853-25mg
3

125,90US$

188,90US$
Guardar 63,00 US$ (33.35%)
100mg
E126853-100mg
3

319,90US$

479,90US$
Guardar 160,00 US$ (33.34%)
500mg
E126853-500mg
2

1.199,90US$

1.799,90US$
Guardar 600,00 US$ (33.34%)
Enter a quantity for the sizes you want to add.
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Why this grade

Moligand™, ≥99% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

🌡

Storage & shipping

Store at -20°C,Argon charged Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

📚

Literature proof

Cited in 37 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Descripción general

Erastin is a cell-permeable piperazinyl-quinazolinone. It interacts with antiporter system Xc-.


Application:

Erastin has been used:
as a positive control for inducing ferroptosis in hepatic stellate cell (HSC)
to induce ferroptosis and in transferrin internalization assay of human fibrosarcoma HT1080 cells
to induce ferroptosis of muscle-derived cell lines

Specifications

Sinónimos
2-(1-(4-(2-(4-chlorophenoxy)acetyl)piperazin-1-yl)ethyl)-3-(2-ethoxyphenyl)quinazolin-4(3H)-one | MFCD09837984 | 2-[1-[4-[2-(4-chlorophenoxy)acetyl]-1-piperazinyl]ethyl]-3-(2-ethoxyphenyl)-4(3H)-Quinazolinone | 2-(1-(4-(2-(4-Chlorophenoxy)acetyl)-1-pipera
Especificaciones y pureza
Moligand™, ≥99%
Mecanismos bioquímicos y fisiológicos
Description:IC50 Value: 0.1 uM (VDAC-2) [1]Erastin is a compound that interacts with VDAC, blocked and reversed mitochondrial depolarization after microtubule destabilizers in intact cells and antagonized tubulin-induced VDAC blockage in planar bilayers.V
Condiciones de almacenamiento de almacenamiento
Store at -20°C, Argon charged
Enviado en
Ice chest + Ice pads
Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.
Grado
Moligand™
Nota
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Pureza
≥99%
Nombres e identificadores
Pubchem Sid504766167
Pubchem Sid Urlhttps://pubchem.ncbi.nlm.nih.gov/substance/504766167
Sonrisas canónicasCCOC1=CC=CC=C1N2C(=O)C3=CC=CC=C3N=C2C(C)N4CCN(CC4)C(=O)COC5=CC=C(C=C5)Cl
IUPAC Name2-[1-[4-[2-(4-chlorophenoxy)acetyl]piperazin-1-yl]ethyl]-3-(2-ethoxyphenyl)quinazolin-4-one
InChIKeyBKQFRNYHFIQEKN-UHFFFAOYSA-N
INCHI1S/C30H31ClN4O4/c1-3-38-27-11-7-6-10-26(27)35-29(32-25-9-5-4-8-24(25)30(35)37)21(2)33-16-18-34(19-17-33)28(36)20-39-23-14-12-22(31)13-15-23/h4-15,21H,3,16-20H2,1-2H3
Isómeros SMILES CCOC1=CC=CC=C1N2C(=O)C3=CC=CC=C3N=C2C(C)N4CCN(CC4)C(=O)COC5=CC=C(C=C5)Cl
WGK Alemania 3
Peso molecular 547.04
Reaxy-Rn 14580272
Reaxys-RN_link_address https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=14580272&ln=

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Taxonomic Classification

Taxonomy Tree

KingdomOrganic compounds
SuperclassOrganoheterocyclic compounds
ClaseDiazanaphthalenes
SubclassBenzodiazines
Intermediate Tree Nodes Not available
Direct ParentQuinazolines
Alternative Parents Phenoxy compounds  Phenol ethers  Pyrimidones  Alkyl aryl ethers  Aralkylamines  N-alkylpiperazines  Chlorobenzenes  Aryl chlorides  Tertiary carboxylic acid amides  Heteroaromatic compounds  Trialkylamines  Amino acids and derivatives  Lactams  Azacyclic compounds  Organopnictogen compounds  Hydrocarbon derivatives  Organic oxides  Organochlorides  Carbonyl compounds  
Molecular FrameworkAromatic heteropolycyclic compounds
Substituents Quinazoline - Phenoxy compound - Phenol ether - Alkyl aryl ether - Chlorobenzene - Halobenzene - Pyrimidone - N-alkylpiperazine - Aralkylamine - Aryl chloride - Aryl halide - Monocyclic benzene moiety - 1,4-diazinane - Piperazine - Pyrimidine - Benzenoid - Tertiary carboxylic acid amide - Heteroaromatic compound - Amino acid or derivatives - Tertiary aliphatic amine - Tertiary amine - Carboxamide group - Lactam - Azacycle - Carboxylic acid derivative - Ether - Amine - Organic oxygen compound - Organopnictogen compound - Organohalogen compound - Carbonyl group - Hydrocarbon derivative - Organochloride - Organonitrogen compound - Organooxygen compound - Organic oxide - Organic nitrogen compound - Aromatic heteropolycyclic compound
DescripciónThis compound belongs to the class of organic compounds known as quinazolines. These are compounds containing a quinazoline moiety, which is made up of two fused six-member aromatic rings, a benzene ring and a pyrimidine ring.
External Descriptors Not available
Estructura 3D
Modelo de Estructura Química Interactiva





Objetivos asociados (humanos)
SLC7A11 Tchem Cystine/glutamate transporter (3 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
VDAC2 Tchem Voltage-dependent anion-selective channel protein 2 (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
A673 (619 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Calu-1 (518 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HL-60 (67320 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HT-1080 (3966 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SK-N-MC (815 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
U2OS (164939 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
U-937 (7138 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
A549 (127892 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
BJ (6930 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
MIA PaCa-2 (5949 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HCT-116 (91556 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HOS (906 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HepG2 (196354 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SK-ES1 (32 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
LNCaP (8286 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HeLa (62764 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Liver (3974 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
VDAC2 Tchem Voltage-dependent anion-selective channel protein 2 (5 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SLC7A11 Tchem Cystine/glutamate transporter (150 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
MAPK3 Tchem Mitogen-activated protein kinase; ERK1/ERK2 (651 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SK-LMS-1 (121 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SW982 (212 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SJSA-1 (970 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SW872 (162 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
C-33-A (287 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Objetivos asociados (no humanos)
Hdac6 Histone deacetylase 6 (222 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
SVR (53 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
rep Replicase polyprotein 1ab (378 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Mecanismos de acción
Certificados (CoA, COO, BSE/TSE y tabla de análisis)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:

Find and download the COA for your product by matching the lot number on the packaging.

21 results found

Lot NumberCertificate TypeFechaArticulo
L2205573Certificate of AnalysisJun 09, 2026 E126853
L2205572Certificate of AnalysisJun 09, 2026 E126853
G2524060Certificate of AnalysisAug 01, 2025 E126853
H2525471Certificate of AnalysisJul 30, 2025 E126853
H2525470Certificate of AnalysisJul 30, 2025 E126853
H2525469Certificate of AnalysisJul 30, 2025 E126853
H2525468Certificate of AnalysisJul 30, 2025 E126853
H2328430Certificate of AnalysisJun 10, 2025 E126853
H2328432Certificate of AnalysisJun 10, 2025 E126853
G2430349Certificate of AnalysisJun 21, 2024 E126853
G2430350Certificate of AnalysisJun 21, 2024 E126853
G2430351Certificate of AnalysisJun 21, 2024 E126853
C2426003Certificate of AnalysisAug 10, 2023 E126853
H2328431Certificate of AnalysisAug 10, 2023 E126853
L2205441Certificate of AnalysisNov 22, 2022 E126853
L2205576Certificate of AnalysisNov 22, 2022 E126853
F2209177Certificate of AnalysisMay 19, 2022 E126853
F2209175Certificate of AnalysisMay 19, 2022 E126853
F2209128Certificate of AnalysisMay 19, 2022 E126853
F2209101Certificate of AnalysisMay 19, 2022 E126853
C2221030Certificate of AnalysisMar 24, 2022 E126853

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Propiedades químicas y físicas
Solubilidad25°C: DMSO
Sensibilidadair & heat sensitive
Peso molecular547.000 g/mol
XLogP34.800
Hydrogen Bond Donor Count0
Hydrogen Bond Acceptor Count6
Rotatable Bond Count8
Exact Mass546.203 Da
Monoisotopic Mass546.203 Da
Topological Polar Surface Area74.700 Ų
Heavy Atom Count39
Formal Charge0
Complexity871.000
Isotope Atom Count0
Defined Atom Stereocenter Count0
Undefined Atom Stereocenter Count1
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
The total count of all stereochemical bonds0
Covalently-Bonded Unit Count1
Preguntas frecuentes y artículos
Citations of This Product
Referencias
1. Junwei Liu, Meihong Zhang, Chuanbin Wu, Xin Pan, Zhengwei Huang.  (2023)  TPGS/soluplus® blended micelles: an effective strategy for improving loading capacity of ferroptosis inducer erastin.  JOURNAL OF DISPERSION SCIENCE AND TECHNOLOGY,      [PMID:] [10.1080/01932691.2023.2295024]
2. Qiang-Ming Li, Tong Xu, Xue-Qiang Zha, Xiao-Wen Feng, Feng-Yun Zhang, Jian-Ping Luo.  (2023)  Buddlejasaponin IVb ameliorates ferroptosis of dopaminergic neuron by suppressing IRP2-mediated iron overload in Parkinson's disease.  JOURNAL OF ETHNOPHARMACOLOGY,      [PMID:37717841] [10.1016/j.jep.2023.117196]
3. Jiangbo Nie, Yuhang Ling, Mingchao Jin, Zhuo Chen, Wei Liu, Weiyun Shen, Tianshun Fang, Jianyou Li, Ying He.  (2023)  Butyrate enhances erastin-induced ferroptosis of osteosarcoma cells via regulating ATF3/SLC7A11 pathway.  EUROPEAN JOURNAL OF PHARMACOLOGY,      [PMID:37619784] [10.1016/j.ejphar.2023.176009]
4. Xinmei Wang, Shanshan Li, Jiayu Yu, Wenlin Wang, Zhuoqi Du, Shuchun Gao, Yin Ma, Ruixin Tang, Ting Liu, Shiping Ma, Qiang Fu, Xueyang Deng.  (2023)  Saikosaponin B2 ameliorates depression-induced microglia activation by inhibiting ferroptosis-mediated neuroinflammation and ER stress.  JOURNAL OF ETHNOPHARMACOLOGY,      [PMID:37277081] [10.1016/j.jep.2023.116729]
5. Xinyu Zhang, Xueli Xu, Huimin Liu, Nengyi Ni, Shuangqing Liu, Yufang Gong, Guiqi Ma, Linlin Song, Qingwei Meng, Qing Fan, Xiao Sun.  (2023)  CCR2-overexpressing biomimetic carrier-free nanoplatform for enhanced cascade ferroptosis tumor therapy.  Acta Biomaterialia,      [PMID:37156432] [10.1016/j.actbio.2023.05.006]
6. Huang Hui, Ye Zhifang, Li Zhengzhao, Wang Bo, Li Ke, Zhou Kai, Cao Huiyuan, Zheng Jiaxuan, Wang Guangji.  (2023)  Employing machine learning using ferroptosis-related genes to construct a prognosis model for patients with osteosarcoma.  Frontiers in Genetics,      [PMID:36733341] [10.3389/fgene.2023.1099272]
7. Jing Zhao, Mingming Ma, Lei Li, Gaoli Fang.  (2023)  Oxysophoridine protects against cerebral ischemia/reperfusion injury via inhibition of TLR4/p38MAPK‑mediated ferroptosis.  Molecular Medicine Reports,  27  (2): (1-11).  [PMID:36601753] [10.3892/mmr.2023.12931]
8. Feng-guo Zhai, Qi-chao Liang, Yi-yan Wu, Jia-qi Liu, Jia-wei Liu.  (2022)  Red ginseng polysaccharide exhibits anticancer activity through GPX4 downregulation-induced ferroptosis.  PHARMACEUTICAL BIOLOGY,      [PMID:35575436] [10.1080/13880209.2022.2066139]
9. Xiazhen Bao, Xuehui Cao, Yong Yuan, Bo Zhou, Congde Huo.  (2021)  A water-soluble, highly sensitive and ultrafast fluorescence probe for imaging of mitochondrial hypochlorous acid.  SENSORS AND ACTUATORS B-CHEMICAL,      [PMID:] [10.1016/j.snb.2021.130210]
10. Na Wei, Tan Lu, Libin Yang, Yonghan Dong, Xiaotan Liu.  (2021)  Lipoxin A4 protects primary spinal cord neurons from Erastin-induced ferroptosis by activating the Akt/Nrf2/HO-1 signaling pathway.  FEBS Open Bio,  11  (8): (2118-2126).  [PMID:34048148] [10.1002/2211-5463.13203]
11. Zhu Yiming, Zhang Chihao, Huang Mingzhe, Lin Jiayun, Fan Xiao, Ni Tao.  (2021)  TRIM26 Induces Ferroptosis to Inhibit Hepatic Stellate Cell Activation and Mitigate Liver Fibrosis Through Mediating SLC7A11 Ubiquitination.  Frontiers in Cell and Developmental Biology,      [PMID:33869196] [10.3389/fcell.2021.644901]
12. Guo-qiang Liang, Wei Mu, Chun-bo Jiang.  (2024)  Baicalein improves renal interstitial fibrosis by inhibiting the ferroptosis in vivo and in vitro.  Heliyon,      [PMID:38601597] [10.1016/j.heliyon.2024.e28954]
13. Zi-Han Xu, Ming-Min Xie, Chun-Lan Xie, Xian-Wen Yang, Jun-Song Wang.  (2025)  Deep-Sea-Derived Isobisvertinol Targets TLR4 to Exhibit Neuroprotective Activity via Anti-Inflammatory and Ferroptosis-Inhibitory Effects.  Marine Drugs,  23  (1): (49).  [PMID:39852551] [10.3390/md23010049]
14. Jie Jiang, Yuqing Gao, Jiang Wang, Yan Huang, Rong Yang, Yongxin Zhang, Yuandi Ma, Yingquan Wen, Gongkai Luo, Shurui Zhang, Yutang Cao, Minjun Yu, Qinxue Wang, Shulei Hu, Kanglong Wang, Xiaozhen Guo, Frank J. Gonzalez, Yameng Liu, Hong Liu, Qing Xie, Cen Xie.  (2025)  Hepatic sphingomyelin phosphodiesterase 3 promotes steatohepatitis by disrupting membrane sphingolipid metabolism.  Cell Metabolism,      [PMID:40015281] [10.1016/j.cmet.2025.01.016]
15. Chen Kechun, Xu Bingtian, Long Lu, Wen Huizhen, Zhao Qian, Tu Xingxing, Wang Jiakang, Xu Jiangping, Wang Haitao.  (2024)  Inhibition of Phosphodiesterase 4 Suppresses Neuronal Ferroptosis After Cerebral Ischemia/Reperfusion.  MOLECULAR NEUROBIOLOGY,      [PMID:39287745] [10.1007/s12035-024-04495-9]
16. Zhou Hao, Wang Wei, Cai Zedong, Jia Zhou-Yan, Li Yu-Yao, He Wei, Li Chen, Zhang Bang-Le.  (2024)  Injectable hybrid hydrogels enable enhanced combination chemotherapy and roused anti-tumor immunity in the synergistic treatment of pancreatic ductal adenocarcinoma.  JOURNAL OF NANOBIOTECHNOLOGY,  22  (1): (1-21).  [PMID:38902759] [10.1186/s12951-024-02646-7]
17. Yu Fu, Guiqin Huang, Yawen Cai, Menghui Ren, Run Cheng, Yuhui Chai, Yingdi Wang, Yunqi An, Tianhua Yan, Lingpeng Zhu, Xinxin Liu.  (2025)  Integrated network pharmacology, bioinformatics, and experiment analysis to decipher the molecular mechanism of Salidroside on Gastric cancer via targeting NCOA4-mediated ferritinophagy.  CHEMICO-BIOLOGICAL INTERACTIONS,      [PMID:39746501] [10.1016/j.cbi.2024.111368]
18. Tang Yuan-juan, Zhang Zhen, Yan Tong, Chen Ken, Xu Guo-fan, Xiong Shi-qiang, Wu Dai-qian, Chen Jie, Jose Pedro A., Zeng Chun-yu, Fu Jin-juan.  (2024)  Irisin attenuates type 1 diabetic cardiomyopathy by anti-ferroptosis via SIRT1-mediated deacetylation of p53.  Cardiovascular Diabetology,  23  (1): (1-19).  [PMID:38566123] [10.1186/s12933-024-02183-5]
19. Kunyi Zhao, Bo Lin, Ling Ma, Qi Zan, Rui Wang, Ruijin Li, Yu Wang, Shaomin Shuang, Chuan Dong, Li Fan.  (2024)  Lipid droplet-targetable fluorescent probe for imaging viscosity in PM2.5 exposure-induced lung injury, non-alcoholic fatty liver, and tumor models.  MICROCHEMICAL JOURNAL,      [PMID:] [10.1016/j.microc.2024.111193]
20. Su Borui, Gao Dong, Xin Nini, Wu Kai, Yang Mei, Jiang Shichao, Zhang Yusheng, Ding Jie, Wu Chengheng, Sun Jing, Wei Dan, Fan Hongsong, Guo Zhenzhen.  (2024)  Mild Synthesis of Ultra-Bright Carbon Dots with Solvatochromism for Rapid Lipid Droplet Monitoring in Varied Physiological Process.  Regenerative Biomaterials,      [PMID:38404618] [10.1093/rb/rbad109]
21. Yilin Pi, Huaiwen Zuo, Yuxin Wang, Weiping Zheng, Huiyuan Zhou, Lamei Deng, Hongli Song.  (2024)  Oleanolic acid alleviating ischemia-reperfusion injury in rat severe steatotic liver via KEAP1/NRF2/ARE.  INTERNATIONAL IMMUNOPHARMACOLOGY,      [PMID:38972213] [10.1016/j.intimp.2024.112617]
22. Cong Lili, Shen Yanting, Wang Jiaqi, Meng Fanxiang, Xu Weiqing, Sun Weixia, Xu Shuping.  (2024)  Revealing mitochondrial microenvironmental changes triggered by ferroptosis regulation.  ANALYTICAL AND BIOANALYTICAL CHEMISTRY,      [PMID:39535559] [10.1007/s00216-024-05638-6]
23. Guiqin Huang, Yawen Cai, Menghui Ren, Xiaoyu Zhang, Yu Fu, Run Cheng, Yingdi Wang, Mingxing Miao, Lingpeng Zhu, Tianhua Yan.  (2024)  Salidroside sensitizes Triple-negative breast cancer to ferroptosis by SCD1-mediated lipogenesis and NCOA4-mediated ferritinophagy.  Journal of Advanced Research,      [PMID:39353532] [10.1016/j.jare.2024.09.027]
24. Haonan Tang, Xiao Zhou, Lijuan Liu, Ziyu Wang, Chen Wang, Ningbin Luo, Guanqiao Jin.  (2024)  Superparamagnetic Iron Oxide–Erastin–Polyethylene Glycol Nanotherapeutic Platform: A Ferroptosis-Based Approach for the Integrated Diagnosis and Treatment of Nasopharyngeal Cancer.  MOLECULAR PHARMACEUTICS,      [PMID:38736196] [10.1021/acs.molpharmaceut.3c01172]
25. Tianfeng Yang, Suyu Zhang, Kun Nie, Xiuhong Peng, Jian Huo, Xiao Fu, Yanmin Zhang.  (2025)  WWOX-mediated p53/SAT1 and NRF2/FPN1 axis contribute to toosendanin-induced ferroptosis in hepatocellular carcinoma.  BIOCHEMICAL PHARMACOLOGY,      [PMID:39894307] [10.1016/j.bcp.2025.116790]
26. Wenhui Liu, Ruyu Cao, Yongye Shen, Yaxin Lu, Shuqi Li, Shen Li, Guochen Su, Jing Xu, Yuanqiang Guo.  (2025)  A TME-responsive polysaccharide nanoplatform integrating synergetic therapy for cancer.  INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES,      [PMID:40858170] [10.1016/j.ijbiomac.2025.147113]
27. Yang Tang, Zheng Wang, Feng Zhou, Ling Li, Chen Sun, Linhui Li, Fei Tang, Dongqin Huang, Zewei Li, Yang Tan, Gang Pei.  (2025)  Benzoylpaeoniflorin alleviates ulcerative colitis by inhibiting ferroptosis through targeting phosphogluconic dehydrogenase.  PHYTOMEDICINE,      [PMID:40829505] [10.1016/j.phymed.2025.157111]
28. Huimei Zhao, Haiyan Zhang, Jianyu Shi, Yanru Liu, Jingao Yu, Yuangui Yang, Jingyu Weng, Zhongxing Song, Rui Zhou, Hong Min, Jian Yao, Mei Wang, Zhen Zhang.  (2025)  Wuwei Shaji powder alleviates OVA-induced allergic asthma by protecting bronchial epithelial cells from ferroptosis via the S-sulfhydration of Keap1.  JOURNAL OF ETHNOPHARMACOLOGY,      [PMID:40222689] [10.1016/j.jep.2025.119649]
29. Zhong He, Hui Long, Hongyue Ma, Wanrong Ran, Yinhong Song, Wenjuan Shang, Junhui Wang, Ye Qin, Zhangshuang Deng.  (2025)  4, 9-dihydroxy-α-lapachone as a potent antiproliferation agent for triple-negative breast cancer via ferroptosis.  FITOTERAPIA,      [PMID:40280251] [10.1016/j.fitote.2025.106567]
30. Song Chao, Shen Baoxin, Chen Chaoqi, Yang Lei, Zhang Chi, Liu Fei, Chen Feng, Wu Xiaofei.  (2025)  Identification of ferroptosis-related genes and potential drugs in osteoarthritis.  INFLAMMATION RESEARCH,  74  (1): (1-20).  [PMID:40299032] [10.1007/s00011-025-02040-5]
31. Lishan Lin, Danhui Huang, Haohua Huang, Lingyan Xie, Yi Huang, Cuiping Ye, Lanhe Chu, Yujie Qiao, Xiaojing Meng, Shaoxi Cai, Hangming Dong.  (2025)  Lung microbiota metabolite L-malic acid attenuates the airway inflammation in asthma by inhibiting ferroptosis.  TOXICOLOGY AND APPLIED PHARMACOLOGY,      [PMID:40381742] [10.1016/j.taap.2025.117396]
32. Weng Xiuhong, Wang Simin, Wang Qing, Wei Mingbo, Cheng Bo.  (2025)  Melatonin inhibits salivary gland epithelial cell ferroptosis via the NRF2/HO-1/GPX4 signaling pathway in primary Sjögren’s syndrome.  INFLAMMATION RESEARCH,  74  (1): (1-19).  [PMID:40413364] [10.1007/s00011-025-02047-y]
33. Junhui Yu, Ningning Shao, Jianming Yang, Long Yang, Kaiwen Hong, Yuzhu Chen, Xiaoming Zhao, Hongzhi Yu, Tao Zhang, Jinrui Dong.  (2025)  Ultrafine garlic powder alleviates non-alcoholic steatohepatitis by inhibiting hepatocyte ferroptosis and modulating ERK-dependent oxidative stress.  Frontiers in Pharmacology,      [PMID:41347177] [10.3389/fphar.2025.1711917]
34. Mengdi Cui, Yi An, Jingling Zhao, Miaoxin Hui, Zhili Xiong, Bing Guan, Yinfeng Shen, Yinshui Zou, Chengyin Li, Rui Wang.  (2025)  Dahuang Gancao Decoction Suppresses Ferroptosis via SIRT3-Mediated NRF2 Deacetylation in Acute Kidney Injury.  PHYTOMEDICINE,      [PMID:41447840] [10.1016/j.phymed.2025.157724]
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