The Calcium-sensing receptor (CaSR) is a class C G protein-coupled receptor that is activated by extracellular calcium ions. It is expressed in various tissues, including the parathyroid gland, thyroid gland, kidney, and bone . The CaSR plays a crucial role in the regulation of calcium homeostasis and bone metabolism.
Calcium-sensing receptor
- NPS-2143, Allosteric modulator of CaS receptor;Allosteric modulator of GPRC6 receptor;Allosteric modulator of mGlu 5 receptor
Cas#:284035-33-2
Starting at $58.90
- Cinacalcet, Allosteric modulator of CaS receptor;Allosteric modulator of mGlu 5 receptor
Cas#:226256-56-0
Starting at $30.90
- 1-arylmethylpyrrolidin-2-yl ethanol amine, Antagonist of CaS receptor
Starting at $1,334.90
- 2-methyl-3-phenethyl-3H-pyrimidin-4-one, Antagonist of CaS receptor
Starting at $1,300.90
- calindol, Allosteric modulator of CaS receptor;Allosteric modulator of GPRC6 receptor
Cas#:374933-30-9
Starting at $1,334.90
- evocalcet, Calcium sensing receptor positive allosteric modulator
Cas#:870964-67-3
Starting at $1,334.90