Leukotriene receptors are a class of G protein-coupled receptors that are activated by leukotrienes, a group of eicosanoid inflammatory mediators that are produced in response to injury or infection. There are two known leukotriene receptors: LTB4 receptor 1 (BLT1) and cysteinyl leukotriene receptor 1 (CysLT1).
Leukotriene receptors
- MK 571, Antagonist of CysLT 1 receptor
Cas#:115104-28-4
- Gue 1654, Allosteric modulator of OXE receptor
Cas#:397290-30-1
- LY223982, Antagonist of BLT 1 receptor
Cas#:117423-74-2
- SR 2640 hydrochloride, Antagonist of CysLT 1 receptor
Cas#:105350-26-3
- 15(S)-HETE, Agonist of BLT 2 receptor
Cas#:54845-95-3
- U-75302, Antagonist of BLT 1 receptor
Cas#:119477-85-9
- 5-OxoETE, Agonist of OXE receptor
Cas#:106154-18-1
- 20-OH-LTB4, Agonist of BLT 1 receptor
Cas#:79516-82-8
- 12-epi Leukotriene B4, Agonist of BLT 2 receptor
Cas#:83709-73-3
- 12(R)-HETE, Agonist of BLT 1 receptor
Cas#:82337-46-0
- 5-oxo-ODE, Agonist of OXE receptor
Cas#:1021188-25-9
- 5-oxo-15-HETE, Agonist of OXE receptor
Cas#:142828-12-4
- CP-195543, Leukotriene B4 receptor antagonist
Cas#:204981-48-6
- CP105696, Antagonist of BLT 1 receptor
Cas#:158081-99-3
- ICI198615, Antagonist of CysLT 1 receptor
Cas#:104448-53-5