Endothelin receptors are a class of G protein-coupled receptors that are activated by endothelin, a peptide hormone that is involved in the regulation of various physiological processes, including blood pressure, vascular tone, and cell proliferation. There are two main types of endothelin receptors: endothelin receptor type A (ETA) and endothelin receptor type B (ETB).
Endothelin receptors
- BQ-123, Antagonist of ET A receptor
Cas#:136553-81-6
- RE 201, Type-1 angiotensin II receptor antagonist
Cas#:254740-64-2
- Avosentan, Endothelin receptor ET-A antagonist
Cas#:290815-26-8
- Macitentan, Endothelin receptor, ET-A/ET-B antagonist
Cas#:441798-33-0
- FR 139317, Antagonist of ET A receptor
Cas#:142375-60-8
- BQ-3020 TFA salt, Agonist of ET B receptor
Cas#:143113-45-5(free basis)
- Bosentan, Endothelin receptor, ET-A/ET-B antagonist
Cas#:147536-97-8
- IRL-2500, Antagonist of ET B receptor
Cas#:169545-27-1
- Lu-135252, Endothelin receptor ET-B antagonist
Cas#:171714-84-4
- PD 151,242, Antagonist of ET A receptor
Cas#:155561-67-4
- A192621, Antagonist of ET B receptor
Cas#:195529-54-5
- BQ788, Antagonist of ET B receptor
Cas#:173326-37-9
- PD-156707, Antagonist of ET A receptor
Cas#:162412-70-6
- aprocitentan, Endothelin receptor, ET-A/ET-B antagonist
Cas#:1103522-45-7
- endothelin-1, Agonist of ET A receptor
Cas#:123626-67-5
- endothelin-3, Agonist of ET B receptor
Cas#:125692-40-2
- endothelin-2, Agonist of ET A receptor
Cas#:122879-69-0
- Ro 46-8443, Antagonist of ET B receptor
Cas#:175556-12-4
- clazosentan, Endothelin receptor ET-A antagonist
Cas#:180384-56-9