Synthetic organic ligands
We offer a diverse range of synthetic organic ligands tailored for various research and development (R&D) applications. These ligands are meticulously designed and synthesized to meet the specific needs of researchers in fields such as chemistry, biology, pharmacology, and materials science. Our collection includes a wide variety of ligands, ranging from small molecules to complex organic compounds, carefully crafted to target specific receptors, enzymes, or biomolecular interactions. With their exceptional purity, reliability, and versatility, our synthetic organic ligands empower researchers to explore new frontiers in drug discovery, chemical biology, and beyond, driving innovation and advancing scientific knowledge in diverse domains.
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- 3-phosphoinositide dependent protein kinase 1 Inhibitor7item
- 5-HT1A receptor Agonist53item
- 5-HT1A receptor Antagonist36item
- 5-HT1B receptor Agonist39item
- 5-HT1B receptor Antagonist19item
- 5-HT1D receptor Agonist39item
- 5-HT1D receptor Antagonist16item
- 5-ht1e receptor Agonist22item
- 5-ht1e receptor Antagonist6item
- 5-HT1F receptor Agonist21item
- 5-HT2A receptor Agonist35item
- 5-HT2A receptor Antagonist76item
- 5-HT2B receptor Agonist33item
- 5-HT2B receptor Antagonist45item
- 5-HT2C receptor Agonist28item
- 5-HT2C receptor Antagonist47item
- 5-HT3A Agonist7item
- 5-HT3A Antagonist18item
- 5-HT4 receptor Agonist21item
- 5-HT4 receptor Antagonist18item
- 5-HT5A receptor Agonist6item
- 5-HT5A receptor Antagonist6item
- 5-HT6 receptor Agonist23item
- 5-HT6 receptor Antagonist35item
- 5-HT7 receptor Agonist22item
- 5-HT7 receptor Antagonist31item
- A1 receptor Agonist29item
- A1 receptor Antagonist55item
- A2A receptor Agonist29item
- A2A receptor Antagonist55item
- A2B receptor Agonist16item
- A2B receptor Antagonist57item
- A3 receptor Agonist32item
- A3 receptor Antagonist53item
- ABL proto-oncogene 1,non-receptor tyrosine kinase Inhibitor29item
- acetyl-CoA acetyltransferase 1 Inhibitor13item
- Acetyl-CoA carboxylase 2 Inhibitor6item
- acetylcholinesterase (Cartwright blood group) Inhibitor8item
- activin A receptor type 1 Inhibitor11item
- activin A receptor type IL Inhibitor7item
- ADAM17 Inhibitor6item
- AKT serine/threonine kinase 1 Inhibitor14item
- AKT serine/threonine kinase 2 Inhibitor13item
- AKT serine/threonine kinase 3 Inhibitor12item
- aldo-keto reductase family 1 member B Inhibitor6item
- ALK receptor tyrosine kinase Inhibitor25item
- Androgen receptor Antagonist11item
- Angiotensin-converting enzyme Inhibitor31item
- Antibiotic9item
- AP2 associated kinase 1 Inhibitor6item
- apelin receptor Agonist10item
- ASIC1 Channel blocker10item
- ASIC3 Channel blocker7item
- AT1 receptor Antagonist25item
- ATM serine/threonine kinase Inhibitor8item
- ATPase family AAA domain containing 2 Inhibitor6item
- ATR serine/threonine kinase Inhibitor10item
- aurora kinase A Inhibitor36item
- aurora kinase B Inhibitor35item
- aurora kinase C Inhibitor8item
- autotaxin Inhibitor9item
- AXL receptor tyrosine kinase Inhibitor19item
- B-Raf proto-oncogene,serine/threonine kinase Inhibitor24item
- B0AT1 Inhibitor6item
- B1 receptor Antagonist7item
- B2 receptor Antagonist7item
- BB3 receptor Agonist13item
- beta-secretase 1 Inhibitor33item
- beta-secretase 2 Inhibitor18item
- BLK proto-oncogene,Src family tyrosine kinase Inhibitor15item
- BLT1 receptor Antagonist10item
- BMX non-receptor tyrosine kinase Inhibitor11item
- bone morphogenetic protein receptor type IA Inhibitor6item
- bromodomain and PHD finger containing 111item
- bromodomain containing 2 Inhibitor15item
- bromodomain containing 3 Inhibitor11item
- bromodomain containing 4 Inhibitor42item
- bromodomain containing 9 Inhibitor9item
- Bruton tyrosine kinase Inhibitor51item
- BUB1 mitotic checkpoint serine/threonine kinase Inhibitor6item
- c-ros oncogene 1,receptor tyrosine kinase Inhibitor6item
- C5a1 receptor Antagonist8item
- CaCC Channel blocker7item
- carbonic anhydrase 1 Inhibitor11item
- carbonic anhydrase 12 Inhibitor11item
- carbonic anhydrase 14 Inhibitor6item
- carbonic anhydrase 4 Inhibitor6item
- carbonic anhydrase 7 Inhibitor7item
- CaS receptor Allosteric modulator14item
- Casein kinase 2 Inhibitor8item
- cathepsin K Inhibitor11item
- cathepsin L Inhibitor8item
- cathepsin S Inhibitor7item
- Cav1.2 Gating inhibitor6item
- Cav3.1 Channel blocker8item
- Cav3.2 Channel blocker9item
- Cav3.3 Channel blocker8item
- CB1 receptor Agonist16item
- CB1 receptor Antagonist16item
- CB2 receptor Agonist21item
- CB2 receptor Antagonist7item
- CCK1 receptor Antagonist23item
- CCK2 receptor Antagonist28item
- CCR1 Antagonist6item
- CCR2 Antagonist13item
- CCR3 Antagonist12item
- CCR4 Antagonist6item
- CCR5 Antagonist16item
- CDC like kinase 1 Inhibitor7item
- CDC like kinase 2 Inhibitor10item
- CDC like kinase 4 Inhibitor6item
- cell division cycle 7 Inhibitor9item
- cereblon13item
- CFTR Activator12item
- CGRP receptor Antagonist9item
- checkpoint kinase 1 Inhibitor16item
- checkpoint kinase 2 Inhibitor11item
- coactivator associated arginine methyltransferase 1 Inhibitor9item
- coagulation factor II,thrombin Inhibitor8item
- coagulation factor X Inhibitor9item
- colony stimulating factor 1 receptor Inhibitor31item
- CoV 3C-like (main) protease Inhibitor59item
- CoV Papain-like protease Inhibitor8item
- COX-1 Inhibitor14item
- COX-2 Inhibitor21item
- CREB binding protein Inhibitor6item
- CRF1 receptor Antagonist12item
- CXCR2 Antagonist8item
- CXCR3 Antagonist6item
- CXCR4 Antagonist7item
- cyclin dependent kinase 1 Inhibitor46item
- cyclin dependent kinase 19 Inhibitor7item
- cyclin dependent kinase 2 Inhibitor46item
- cyclin dependent kinase 4 Inhibitor37item
- cyclin dependent kinase 5 Inhibitor23item
- cyclin dependent kinase 6 Inhibitor21item
- cyclin dependent kinase 7 Inhibitor16item
- cyclin dependent kinase 8 Inhibitor12item
- cyclin dependent kinase 9 Inhibitor29item
- CYP19A1 Inhibitor7item
- CYP3A4 Inhibitor9item
- CYP5A1 Inhibitor7item
- CysLT1 receptor Antagonist15item
- CysLT2 receptor Antagonist9item
- D1 receptor Agonist14item
- D1 receptor Antagonist10item
- D2 receptor Agonist27item
- D2 receptor Antagonist43item
- D3 receptor Agonist18item
- D3 receptor Antagonist28item
- D4 receptor Agonist10item
- D4 receptor Antagonist30item
- D5 receptor Agonist8item
- D5 receptor Antagonist8item
- DAT Inhibitor11item
- dihydroorotate dehydrogenase (quinone) Inhibitor10item
- dipeptidyl peptidase 4 Inhibitor12item
- dipeptidyl peptidase 8 Inhibitor6item
- diphosphomevalonate decarboxylase Inhibitor12item
- discoidin domain receptor tyrosine kinase 1 Inhibitor12item
- discoidin domain receptor tyrosine kinase 2 Inhibitor9item
- DOT1 like histone lysine methyltransferase Inhibitor6item
- DP1 receptor Agonist16item
- DP1 receptor Antagonist10item
- DP2 receptor Agonist9item
- DP2 receptor Antagonist12item
- dual specificity tyrosine phosphorylation regulated kinase 1A Inhibitor14item
- dual specificity tyrosine phosphorylation regulated kinase 1B Inhibitor6item
- enhancer of zeste 2 polycomb repressive complex 2 subunit Inhibitor15item
- EP1 receptor Agonist12item
- EP1 receptor Antagonist9item
- EP2 receptor Agonist19item
- EP2 receptor Antagonist9item
- EP3 receptor Agonist24item
- EP3 receptor Antagonist11item
- EP4 receptor Agonist20item
- EP4 receptor Antagonist18item
- epidermal growth factor receptor Inhibitor70item
- epoxide hydrolase 2 Inhibitor9item
- Equilibrative nucleoside transporter 1 Inhibitor7item
- erb-b2 receptor tyrosine kinase 2 Inhibitor26item
- erb-b2 receptor tyrosine kinase 4 Inhibitor13item
- Estrogen receptor-α Agonist11item
- Estrogen receptor-α Antagonist16item
- Estrogen receptor-β Agonist8item
- Estrogen receptor-β Antagonist10item
- Estrogen-related receptor-γ Agonist6item
- ETA receptor Antagonist16item
- ETB receptor Antagonist10item
- euchromatic histone lysine methyltransferase 2 Inhibitor8item
- Farnesoid X receptor Agonist11item
- farnesyl diphosphate synthase Inhibitor20item
- Fatty acid amide hydrolase Inhibitor19item
- FFA1 receptor Agonist11item
- FGR proto-oncogene,Src family tyrosine kinase Inhibitor6item
- fibroblast growth factor receptor 1 Inhibitor38item
- fibroblast growth factor receptor 2 Inhibitor17item
- fibroblast growth factor receptor 3 Inhibitor23item
- fibroblast growth factor receptor 4 Inhibitor16item
- Five-Membered Heterocyclic Compounds7item
- FKBP prolyl isomerase 1A Inhibitor6item
- fms related receptor tyrosine kinase 1 Inhibitor32item
- fms related receptor tyrosine kinase 3 Inhibitor56item
- fms related receptor tyrosine kinase 4 Inhibitor31item
- FP receptor Agonist22item
- FPR1 Agonist6item
- FPR2/ALX Agonist11item
- FYN proto-oncogene,Src family tyrosine kinase Inhibitor10item
- GABAA receptor α1 subunit Agonist6item
- GABAA receptor α1 subunit Allosteric modulator16item
- GABAA receptor α2 subunit Agonist6item
- GABAA receptor α2 subunit Allosteric modulator17item
- GABAA receptor α3 subunit Agonist6item
- GABAA receptor α3 subunit Allosteric modulator16item
- GABAA receptor α5 subunit Agonist6item
- GABAA receptor α5 subunit Allosteric modulator19item
- GABAA receptor α6 subunit Allosteric modulator9item
- GABAA receptor ρ1 subunit Antagonist6item
- GABAA receptor ρ2 subunit Antagonist6item
- GABAA receptor ρ3 subunit Antagonist6item
- GABAB receptor Antagonist11item
- GABAB1 Antagonist10item
- GAT1 Inhibitor9item
- geranylgeranyl diphosphate synthase Inhibitor19item
- GluA1 Allosteric modulator8item
- GluA2 Allosteric modulator8item
- GluA2 Antagonist7item
- GluA3 Allosteric modulator8item
- GluA4 Allosteric modulator8item
- Glucocorticoid receptor Agonist26item
- GluK1 Agonist8item
- GluK1 Antagonist8item
- GluN1 Agonist6item
- GluN1 Antagonist11item
- GluN2A Agonist6item
- GluN2A Allosteric modulator6item
- GluN2A Antagonist13item
- GluN2B Agonist6item
- GluN2B Antagonist14item
- GluN2C Antagonist13item
- GluN2D Antagonist12item
- Glycine Receptor (All subtypes) Subunit-specific10item
- glycine receptor α2 subunit Antagonist6item
- glycogen synthase kinase 3 alpha Inhibitor7item
- glycogen synthase kinase 3 beta Inhibitor41item
- GlyT1 Inhibitor12item
- GnRH1 receptor Antagonist11item
- GPCR/G Protein20item
- GPER Agonist7item
- GPR119 Agonist31item
- GPR55 Agonist13item
- GPR84 Agonist9item
- Guanylyl cyclase,α1β1 Activator7item
- H1 receptor Agonist14item
- H1 receptor Antagonist56item
- H2 receptor Agonist6item
- H2 receptor Antagonist14item
- H3 receptor Agonist24item
- H3 receptor Antagonist31item
- H4 receptor Agonist19item
- H4 receptor Antagonist15item
- HCA2 receptor Agonist17item
- HCA3 receptor Agonist7item
- HCN1 Channel blocker7item
- HCN2 Channel blocker6item
- HCN4 Channel blocker6item
- histone deacetylase 1 Inhibitor28item
- histone deacetylase 10 Inhibitor8item
- histone deacetylase 2 Inhibitor21item
- histone deacetylase 3 Inhibitor26item
- histone deacetylase 4 Inhibitor11item
- histone deacetylase 5 Inhibitor14item
- histone deacetylase 6 Inhibitor34item
- histone deacetylase 7 Inhibitor11item
- histone deacetylase 8 Inhibitor21item
- histone deacetylase 9 Inhibitor10item
- hydroxymethylglutaryl-CoA reductase Inhibitor67item
- hydroxysteroid 11-beta dehydrogenase 1 Inhibitor7item
- IL2 inducible T cell kinase Inhibitor8item
- indoleamine 2,3-dioxygenase 1 Inhibitor9item
- inhibitor of nuclear factor kappa B kinase subunit beta Inhibitor7item
- inhibitor of nuclear factor kappa B kinase subunit epsilon Inhibitor10item
- Insulin receptor Inhibitor10item
- Insulin-like growth factor I receptor Inhibitor16item
- interleukin 1 receptor associated kinase 1 Inhibitor6item
- interleukin 1 receptor associated kinase 4 Inhibitor15item
- IP receptor Agonist20item
- Janus kinase 1 Inhibitor52item
- Janus kinase 2 Inhibitor73item
- Janus kinase 3 Inhibitor54item
- KCa2.1 Activator6item
- KCa2.2 Activator9item
- KCa2.3 Activator6item
- KCa3.1 Activator9item
- kinase insert domain receptor Inhibitor82item
- Kir3.2 Gating inhibitor6item
- Kir3.4 Channel blocker9item
- KIT proto-oncogene,receptor tyrosine kinase Inhibitor50item
- KRAS Inhibitor11item
- Kv1.7 Channel blocker6item
- Kv10.1 Channel blocker8item
- Kv11.1 Activator8item
- Kv11.1 Channel blocker9item
- lanosterol synthase Inhibitor16item
- LCK proto-oncogene,Src family tyrosine kinase Inhibitor28item
- leucine rich repeat kinase 2 Inhibitor25item
- LIM domain kinase 1 Inhibitor9item
- LPA1 receptor Agonist6item
- LPA1 receptor Antagonist20item
- LPA2 receptor Agonist8item
- LPA3 receptor Agonist8item
- LPA3 receptor Antagonist9item
- LYN proto-oncogene,Src family tyrosine kinase Inhibitor10item
- lysine demethylase 1A Inhibitor7item
- M1 receptor Agonist27item
- M1 receptor Allosteric modulator22item
- M1 receptor Antagonist42item
- M2 receptor Agonist19item
- M2 receptor Allosteric modulator15item
- M2 receptor Antagonist45item
- M3 receptor Agonist19item
- M3 receptor Antagonist37item
- M4 receptor Agonist19item
- M4 receptor Allosteric modulator11item
- M4 receptor Antagonist39item
- M5 receptor Agonist13item
- M5 receptor Antagonist30item
- MAPK activated protein kinase 2 Inhibitor7item
- MCH1 receptor Antagonist15item
- mechanistic target of rapamycin kinase Inhibitor43item
- MER proto-oncogene,tyrosine kinase Inhibitor15item
- MET proto-oncogene,receptor tyrosine kinase Inhibitor39item
- Metabolic Enzyme/Protease11item
- mGlu1 receptor Agonist6item
- mGlu1 receptor Allosteric modulator61item
- mGlu1 receptor Antagonist10item
- mGlu2 receptor Agonist10item
- mGlu2 receptor Allosteric modulator31item
- mGlu2 receptor Antagonist7item
- mGlu3 receptor Agonist7item
- mGlu3 receptor Allosteric modulator10item
- mGlu4 receptor Agonist10item
- mGlu4 receptor Allosteric modulator20item
- mGlu5 receptor Agonist12item
- mGlu5 receptor Allosteric modulator80item
- mGlu5 receptor Antagonist7item
- mGlu6 receptor Agonist11item
- mGlu6 receptor Antagonist6item
- mGlu7 receptor Agonist7item
- mGlu7 receptor Allosteric modulator7item
- mGlu7 receptor Antagonist7item
- mGlu8 receptor Agonist10item
- Mineralocorticoid receptor Antagonist10item
- mitogen-activated protein kinase 1 Inhibitor12item
- mitogen-activated protein kinase 10 Inhibitor12item
- mitogen-activated protein kinase 14 Inhibitor27item
- mitogen-activated protein kinase 7 Inhibitor6item
- mitogen-activated protein kinase 8 Inhibitor11item
- mitogen-activated protein kinase 9 Inhibitor8item
- mitogen-activated protein kinase kinase 1 Inhibitor12item
- mitogen-activated protein kinase kinase kinase 7 Inhibitor9item
- MMP13 Inhibitor8item
- MMP9 Inhibitor7item
- Monoacylglycerol lipase Inhibitor8item
- motilin receptor Agonist10item
- MT1 receptor Agonist26item
- MT2 receptor Agonist30item
- MT2 receptor Antagonist12item
- NET Inhibitor26item
- Neuronal NOS Inhibitor7item
- neurotrophic receptor tyrosine kinase 1 Inhibitor25item
- neurotrophic receptor tyrosine kinase 2 Inhibitor11item
- neurotrophic receptor tyrosine kinase 3 Inhibitor11item
- Neutral endopeptidase Inhibitor12item
- nicotinic acetylcholine receptor α7 subunit Agonist10item
- NK1 receptor Antagonist27item
- NK2 receptor Antagonist12item
- NK3 receptor Antagonist17item
- NOP receptor Agonist7item
- NOP receptor Antagonist8item
- NUAK family kinase 1 Inhibitor7item
- OT receptor Antagonist18item
- OX1 receptor Antagonist25item
- OX2 receptor Agonist8item
- OX2 receptor Antagonist27item
- p21 (RAC1) activated kinase 1 Inhibitor7item
- P2X3 Antagonist10item
- P2X4 Antagonist8item
- P2X7 Antagonist12item
- P2Y1 receptor Agonist9item
- P2Y1 receptor Antagonist16item
- P2Y12 receptor Antagonist18item
- P2Y6 receptor Agonist9item
- PAF receptor Antagonist16item
- Peroxisome proliferator-activated receptor-α Agonist24item
- Peroxisome proliferator-activated receptor-β/δ Agonist9item
- Peroxisome proliferator-activated receptor-γ Agonist42item
- Pharmaceutical ingredients12item
- phosphatidylinositol 3-kinase catalytic subunit type 3 Inhibitor12item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha Inhibitor75item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta Inhibitor59item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta Inhibitor70item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma Inhibitor67item
- phosphodiesterase 4A Inhibitor9item
- phosphodiesterase 4B Inhibitor11item
- phosphodiesterase 4D Inhibitor10item
- phosphodiesterase 5A Inhibitor12item
- Pim-1 proto-oncogene,serine/threonine kinase Inhibitor19item
- Pim-2 proto-oncogene,serine/threonine kinase Inhibitor8item
- Pim-3 proto-oncogene,serine/threonine kinase Inhibitor7item
- platelet derived growth factor receptor alpha Inhibitor25item
- platelet derived growth factor receptor beta Inhibitor47item
- polo like kinase 1 Inhibitor12item
- poly(ADP-ribose) polymerase 1 Inhibitor15item
- poly(ADP-ribose) polymerase 2 Inhibitor7item
- Pregnane X receptor Agonist8item
- protein arginine methyltransferase 5 Inhibitor7item
- protein kinase A Inhibitor7item
- protein kinase C alpha Inhibitor8item
- protein kinase C beta Inhibitor9item
- protein kinase C delta Inhibitor7item
- protein kinase,DNA-activated,catalytic subunit Inhibitor13item
- protein tyrosine kinase 2 Inhibitor9item
- Protein Tyrosine Kinase/RTK16item
- Pyrimidines7item
- Raf-1 proto-oncogene,serine/threonine kinase Inhibitor23item
- RAR-related orphan receptor-γ Agonist15item
- receptor interacting serine/threonine kinase 1 Inhibitor27item
- receptor interacting serine/threonine kinase 2 Inhibitor10item
- regulator of G-protein signaling 4 Inhibitor8item
- ret proto-oncogene Inhibitor26item
- Retinoic acid receptor-α Agonist8item
- Retinoic acid receptor-β Agonist7item
- Retinoic acid receptor-γ Agonist10item
- Retinoid X receptor-α Agonist10item
- Rho associated coiled-coil containing protein kinase 1 Inhibitor14item
- Rho associated coiled-coil containing protein kinase 2 Inhibitor17item
- ribosomal protein S6 kinase A1 Inhibitor7item
- S1P1 receptor Agonist31item
- S1P3 receptor Agonist12item
- S1P4 receptor Agonist16item
- S1P5 receptor Agonist16item
- SERT Inhibitor28item
- Six-Membered Heterocyclic Compounds10item
- SMO Antagonist9item
- Sodium/glucose cotransporter 1 Inhibitor12item
- Sodium/glucose cotransporter 2 Inhibitor10item
- sphingosine kinase 1 Inhibitor10item
- sphingosine kinase 2 Inhibitor11item
- spleen associated tyrosine kinase Inhibitor20item
- squalene synthase Inhibitor77item
- SRC proto-oncogene,non-receptor tyrosine kinase Inhibitor28item
- succinate receptor Agonist7item
- TANK binding kinase 1 Inhibitor13item
- tankyrase 2 Inhibitor8item
- tankyrase Inhibitor8item
- tec protein tyrosine kinase Inhibitor9item
- TEK receptor tyrosine kinase Inhibitor10item
- TP receptor Agonist20item
- TP receptor Antagonist20item
- transforming growth factor beta receptor 1 Inhibitor10item
- TRPA1 Activator23item
- TRPC3 Channel blocker10item
- TRPC5 Channel blocker14item
- TRPC6 Channel blocker15item
- TRPM8 Activator14item
- TRPM8 Channel blocker13item
- TRPML3 Activator7item
- TRPV1 Channel blocker15item
- TTK protein kinase Inhibitor11item
- TXK tyrosine kinase Inhibitor8item
- tyrosine kinase 2 Inhibitor40item
- UT receptor Antagonist10item
- V1A receptor Antagonist15item
- V2 receptor Antagonist10item
- VRAC Channel blocker9item
- YES proto-oncogene 1,Src family tyrosine kinase Inhibitor8item
- α1A-adrenoceptor Antagonist28item
- α1B-adrenoceptor Antagonist26item
- α1D-adrenoceptor Agonist11item
- α1D-adrenoceptor Antagonist28item
- α2A-adrenoceptor Agonist9item
- α2A-adrenoceptor Antagonist13item
- α2B-adrenoceptor Agonist7item
- α2B-adrenoceptor Antagonist18item
- α2C-adrenoceptor Agonist7item
- α2C-adrenoceptor Antagonist19item
- β1-adrenoceptor Agonist19item
- β1-adrenoceptor Antagonist30item
- β2-adrenoceptor Agonist25item
- β2-adrenoceptor Antagonist24item
- β3-adrenoceptor Agonist17item
- β3-adrenoceptor Antagonist11item
- δ receptor Agonist21item
- δ receptor Antagonist18item
- κ receptor Agonist29item
- κ receptor Antagonist18item
- μ receptor Agonist25item
- μ receptor Antagonist20item
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Custom Product
Grade
Action Type
- ACTIVATOR212item
- AGONIST1312item
- ALLOSTERIC ANTAGONIST1 item
- ALLOSTERIC MODULATOR440item
- ANTAGONIST1586item
- BINDING AGENT1 item
- BLOCKER25item
- CHANNEL BLOCKER218item
- CHELATING AGENT1 item
- CROSS-LINKING AGENT2item
- DEGRADER1 item
- GATING INHIBITOR40item
- INHIBITOR3053item
- INVERSE AGONIST5item
- MODULATOR19item
- NEGATIVE ALLOSTERIC MODULATOR5item
- NEGATIVE MODULATOR2item
- OPENER2item
- PARTIAL AGONIST11item
- POSITIVE ALLOSTERIC MODULATOR12item
- POSITIVE MODULATOR8item
- STABILISER3item
- SUBSTRATE1 item
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