Welcome to our Approved Ligands section, meticulously curated for the dynamic realm of scientific services and research and development (R&D) in pharmacology, drug discovery, and therapeutic development. Explore our comprehensive collection of high-quality ligands meticulously vetted and approved for various biomedical applications. From small molecules targeting specific receptors and pathways to biologics and antibody-based therapies, our selection includes compounds with proven efficacy and safety profiles, approved by regulatory agencies worldwide. Whether you're conducting preclinical studies, investigating drug mechanisms, or developing novel therapies, our Approved Ligands offer reliability, precision, and regulatory compliance for your scientific services and R&D endeavors. Discover the potential of approved ligands in accelerating your research and development efforts.
Approved Ligands
- Iloprost, Prostanoid IP receptor agonist
Specifications & Purity: ≥97%
CAS No.: 78919-13-8
Starting at $96.90
- Imatinib (STI571), Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of discoidin domain receptor tyrosine kinase 1;Inhibitor of discoidin domain receptor tyrosine kinase 2
Specifications & Purity: ≥99%
CAS No.: 152459-95-5
Starting at $9.90
- Nadolol, Beta-2 adrenergic receptor antagonist
Specifications & Purity: ≥98%
CAS No.: 42200-33-9
Starting at $48.90
- Chidamide impurity, Inhibitor of histone deacetylase 1
Specifications & Purity: 98%
CAS No.: 743420-02-2
Starting at $53.90
- Lenvatinib (E7080), Inhibitor of fms related receptor tyrosine kinase 4;Inhibitor of kinase insert domain receptor
Specifications & Purity: ≥99%
CAS No.: 417716-92-8
Starting at $48.90
- Palonosetron, Antagonist of 5-HT 3A
Specifications & Purity: 98%
CAS No.: 135729-61-2
Starting at $54.90
- Heparin sodium salt, Activator of serpin family C member 1
Specifications & Purity: ≥180 USP units/mg
CAS No.: 9041-08-1
Starting at $137.90
- Hydroxyurea, Ribonucleoside-diphosphate reductase RR1 inhibitor
Specifications & Purity: 98%
CAS No.: 127-07-1
Starting at $19.90
- Nilutamide, Androgen Receptor antagonist
Specifications & Purity: 98%
CAS No.: 63612-50-0
Starting at $96.90
- Carprofen, Cyclooxygenase-2 inhibitor
Specifications & Purity: >98.0%(HPLC)
CAS No.: 53716-49-7
Starting at $68.90
- Neratinib (HKI-272), Receptor protein-tyrosine kinase erbB-4 inhibitor
Specifications & Purity: ≥99%
CAS No.: 698387-09-6
Starting at $19.90
- S-(-)-Carbidopa, Inhibitor of L-Aromatic amino-acid decarboxylase
Specifications & Purity: 98%
CAS No.: 28860-95-9
Starting at $89.90
- 4-aminobutyrate aminotransferase Inhibitor1 item
- 4-hydroxyphenylpyruvate dioxygenase Inhibitor1 item
- 5-HT1A receptor Agonist9item
- 5-HT1A receptor Antagonist3item
- 5-HT1B receptor Agonist6item
- 5-HT1D receptor Agonist6item
- 5-HT1D receptor Antagonist1 item
- 5-ht1e receptor Agonist4item
- 5-HT1F receptor Agonist3item
- 5-HT2A receptor Agonist4item
- 5-HT2A receptor Antagonist18item
- 5-HT2B receptor Agonist2item
- 5-HT2B receptor Antagonist4item
- 5-HT2C receptor Agonist2item
- 5-HT2C receptor Antagonist8item
- 5-HT3A Antagonist6item
- 5-HT3A Channel blocker1 item
- 5-HT3AB Antagonist1 item
- 5-HT4 receptor Agonist2item
- 5-HT4 receptor Antagonist1 item
- 5-HT5A receptor Agonist1 item
- 5-HT5A receptor Antagonist1 item
- 5-HT6 receptor Antagonist11item
- 5-HT7 receptor Agonist3item
- 5-HT7 receptor Antagonist9item
- 5-LOX Inhibitor1 item
- A1 receptor Agonist2item
- A2A receptor Agonist2item
- A2B receptor Agonist2item
- A3 receptor Agonist2item
- ABCC5 Inhibitor1 item
- ABCG2 Inhibitor1 item
- ABL proto-oncogene 1,non-receptor tyrosine kinase Inhibitor5item
- acetylcholinesterase (Cartwright blood group) Inhibitor2item
- Adenosine deaminase Inhibitor1 item
- Adrenergic Receptor1 item
- Alcohol C10-C111 item
- aldo-keto reductase family 1 member B Inhibitor1 item
- ALK receptor tyrosine kinase Inhibitor4item
- alkaloid2item
- Allosteric modulator1 item
- amine oxidase copper containing 3 Inhibitor1 item
- Amitriptyline1 item
- AMY1 receptor Antagonist1 item
- Androgen receptor Agonist1 item
- Androgen receptor Antagonist6item
- Angiotensin-converting enzyme Inhibitor15item
- Anti-inflammatory Ingredients1 item
- Anti-rheumatoid Arthritis Ingredients1 item
- AP2 associated kinase 1 Inhibitor1 item
- Apoptosis3item
- Aryl hydrocarbon receptor Agonist1 item
- ASIC3 Channel blocker2item
- AT1 receptor Antagonist5item
- ATP4A Inhibitor1 item
- B-Raf proto-oncogene,serine/threonine kinase Inhibitor3item
- Basolateral Na-K-Cl symporter Inhibitor2item
- Bcl-2-like 1 Antagonist1 item
- Bcl-2-like 2 Antagonist1 item
- BCL2 apoptosis regulator Antagonist1 item
- Bioactive small molecules (others)1 item
- BLK proto-oncogene,Src family tyrosine kinase Inhibitor2item
- BMP2 inducible kinase Inhibitor1 item
- BMX non-receptor tyrosine kinase Inhibitor2item
- bone morphogenetic protein receptor type 2 Inhibitor1 item
- bromodomain containing 4 Inhibitor2item
- Bruton tyrosine kinase Inhibitor2item
- butyrylcholinesterase Inhibitor1 item
- c-ros oncogene 1,receptor tyrosine kinase Inhibitor1 item
- CaCC Channel blocker1 item
- calcium/calmodulin dependent protein kinase ID Inhibitor1 item
- calcium/calmodulin-dependent protein kinase II gamma subunit Inhibitor1 item
- carbonic anhydrase 1 Activator1 item
- carbonic anhydrase 1 Inhibitor4item
- carbonic anhydrase 12 Inhibitor4item
- carbonic anhydrase 13 Inhibitor1 item
- carbonic anhydrase 14 Inhibitor4item
- carbonic anhydrase 4 Inhibitor3item
- carbonic anhydrase 7 Inhibitor4item
- Carbonyl compound1 item
- CaS receptor Allosteric modulator1 item
- casein kinase 1 epsilon Inhibitor1 item
- Catechol-O-methyltransferase Inhibitor2item
- CatSper1 Activator2item
- CatSper2 Activator2item
- CatSper3 Activator2item
- CatSper4 Activator2item
- Cav1.1 Channel blocker2item
- Cav1.2 Channel blocker2item
- Cav1.2 Gating inhibitor1 item
- Cav1.3 Channel blocker2item
- Cav1.4 Channel blocker2item
- Cav3.1 Channel blocker1 item
- Cav3.2 Channel blocker1 item
- Cav3.3 Channel blocker1 item
- CCR5 Antagonist1 item
- CFTR Activator1 item
- CGRP receptor Antagonist1 item
- coagulation factor II,thrombin Inhibitor1 item
- coagulation factor X Inhibitor4item
- colony stimulating factor 1 receptor Inhibitor2item
- COX-1 Inhibitor5item
- COX-2 Inhibitor8item
- cyclin dependent kinase 19 Inhibitor3item
- cyclin dependent kinase 4 Inhibitor3item
- cyclin dependent kinase 6 Inhibitor2item
- cyclin dependent kinase 8 Inhibitor2item
- cyclin G associated kinase Inhibitor1 item
- CYP11A1 Inhibitor1 item
- CYP11B1 Inhibitor1 item
- CYP11B2 Inhibitor1 item
- CYP19A1 Inhibitor5item
- CYP2C8 Inhibitor1 item
- CYP2J2 Inhibitor1 item
- CYP3A4 Inhibitor1 item
- CysLT1 receptor Antagonist1 item
- Cytochrome P4501 item
- D1 receptor Agonist3item
- D1 receptor Antagonist2item
- D2 receptor Agonist5item
- D2 receptor Antagonist9item
- D3 receptor Agonist4item
- D3 receptor Antagonist5item
- D4 receptor Agonist3item
- D4 receptor Antagonist5item
- D5 receptor Agonist2item
- D5 receptor Antagonist2item
- DAT Inhibitor2item
- dihydroorotate dehydrogenase (quinone) Inhibitor1 item
- Dipeptidase 1 Inhibitor1 item
- dipeptidyl peptidase 4 Inhibitor6item
- dipeptidyl peptidase 8 Inhibitor1 item
- dipeptidyl peptidase 9 Inhibitor1 item
- discoidin domain receptor tyrosine kinase 1 Inhibitor2item
- discoidin domain receptor tyrosine kinase 2 Inhibitor3item
- DNA topoisomerase I Inhibitor1 item
- Dopamine Receptor1 item
- DP1 receptor Agonist2item
- elastase,neutrophil expressed Inhibitor1 item
- ENaCαβγ Channel blocker1 item
- Endogenous Metabolite2item
- enhancer of zeste 2 polycomb repressive complex 2 subunit Inhibitor1 item
- EP1 receptor Agonist2item
- EP2 receptor Agonist3item
- EP3 receptor Agonist3item
- EP4 receptor Agonist3item
- epidermal growth factor receptor Inhibitor8item
- Equilibrative nucleoside transporter 1 Inhibitor2item
- erb-b2 receptor tyrosine kinase 2 Inhibitor4item
- erb-b2 receptor tyrosine kinase 4 Inhibitor3item
- Estrogen receptor-α Agonist6item
- Estrogen receptor-α Antagonist5item
- Estrogen receptor-β Agonist5item
- Estrogen receptor-β Antagonist5item
- Estrogen-related receptor-α Antagonist1 item
- Estrogen-related receptor-β Antagonist1 item
- Estrogen-related receptor-γ Antagonist1 item
- ETA receptor Antagonist4item
- ETB receptor Antagonist2item
- Farnesoid X receptor Agonist2item
- farnesyl diphosphate synthase Inhibitor3item
- fatty acid binding protein 1 Inhibitor1 item
- Ferroptosis1 item
- FES proto-oncogene,tyrosine kinase Inhibitor1 item
- fibroblast growth factor receptor 1 Inhibitor5item
- fibroblast growth factor receptor 2 Inhibitor2item
- fibroblast growth factor receptor 3 Inhibitor2item
- fibroblast growth factor receptor 4 Inhibitor2item
- FKBP prolyl isomerase 1A Inhibitor3item
- fms related receptor tyrosine kinase 1 Inhibitor5item
- fms related receptor tyrosine kinase 3 Inhibitor5item
- fms related receptor tyrosine kinase 4 Inhibitor7item
- FP receptor Agonist3item
- FPR1 Antagonist2item
- FSH receptor Agonist1 item
- FYN proto-oncogene,Src family tyrosine kinase Inhibitor3item
- fyn related Src family tyrosine kinase Inhibitor1 item
- G-protein coupled receptor1 item
- GABAA receptor α6 subunit Allosteric modulator1 item
- GABAB receptor Agonist1 item
- GAT1 Inhibitor1 item
- GCGR1 item
- GLP-1 receptor Agonist4item
- glucagon receptor Agonist1 item
- Glucocorticoid receptor Agonist13item
- Glucosamine1 item
- Glycine Receptor (All subtypes) Antagonist2item
- Glycine Receptor (All subtypes) Subunit-specific4item
- glycine receptor α1 subunit Antagonist2item
- glycine receptor α2 subunit Antagonist2item
- glycine receptor β subunit Antagonist1 item
- glycogen synthase kinase 3 beta Inhibitor1 item
- GnRH1 receptor Agonist1 item
- GnRH1 receptor Antagonist1 item
- GPBA receptor Agonist1 item
- GPCR/G Protein3item
- GPER Agonist3item
- GPR17 Antagonist1 item
- GPR35 Agonist2item
- H1 receptor Agonist1 item
- H1 receptor Antagonist22item
- H2 receptor Antagonist3item
- H3 receptor Antagonist1 item
- H4 receptor Antagonist1 item
- HCK proto-oncogene,Src family tyrosine kinase Inhibitor1 item
- HDAC1 item
- Hepatitis C virus genome polyprotein Inhibitor1 item
- Histamine receptor antagonists1 item
- histone deacetylase 1 Inhibitor3item
- histone deacetylase 10 Inhibitor1 item
- histone deacetylase 11 Inhibitor1 item
- histone deacetylase 2 Inhibitor2item
- histone deacetylase 3 Inhibitor2item
- histone deacetylase 4 Inhibitor1 item
- histone deacetylase 5 Inhibitor2item
- histone deacetylase 6 Inhibitor2item
- histone deacetylase 7 Inhibitor1 item
- histone deacetylase 8 Inhibitor2item
- histone deacetylase 9 Inhibitor2item
- hydroxy-delta-5-steroid dehydrogenase,3 beta- and steroid delta-isomerase 2 Inhibitor1 item
- hydroxymethylglutaryl-CoA reductase Inhibitor1 item
- IL2 inducible T cell kinase Inhibitor2item
- Immunosuppressant Ingredients1 item
- IMPase 1 Inhibitor1 item
- inhibitor1 item
- Inorganic metal2item
- inosine monophosphate dehydrogenase 1 Inhibitor1 item
- inosine monophosphate dehydrogenase 2 Inhibitor1 item
- Insulin receptor Inhibitor2item
- Insulin-like growth factor I receptor Inhibitor2item
- integrin αIIbβ3 Inhibitor1 item
- integrin,alpha L subunit (antigen CD11A (p180),lymphocyte function-associated antigen 1; alpha polypeptide) Antagonist1 item
- IP receptor Agonist2item
- isocitrate dehydrogenase (NADP(+)) 1 Inhibitor1 item
- JAK1 item
- JAK/STAT Signaling1 item
- Janus kinase 1 Allosteric modulator1 item
- Janus kinase 1 Inhibitor7item
- Janus kinase 2 Inhibitor7item
- Janus kinase 3 Inhibitor9item
- K2P10.1 Activator1 item
- K2P12.1 Inhibitor1 item
- K2P13.1 Inhibitor1 item
- K2P2.1 Activator1 item
- K2P3.1 Activator1 item
- K2P5.1 Activator1 item
- K2P9.1 Activator1 item
- Kidney-specific Na-K-Cl symporter Inhibitor2item
- kinase insert domain receptor Inhibitor13item
- Kir3.2 Channel blocker2item
- Kir3.2 Gating inhibitor4item
- Kir3.4 Activator1 item
- Kir3.4 Channel blocker2item
- KIT proto-oncogene,receptor tyrosine kinase Inhibitor4item
- KNa1.1 Activator1 item
- Kv1.1 Channel blocker2item
- Kv1.2 Channel blocker2item
- Kv1.5 Channel blocker2item
- Kv1.7 Channel blocker3item
- Kv1.8 Channel blocker2item
- Kv10.1 Channel blocker3item
- Kv11.1 Channel blocker4item
- Kv2.1 Channel blocker1 item
- Kv3.1 Channel blocker2item
- Kv3.1 Gating inhibitor1 item
- Kv3.2 Channel blocker1 item
- L-Aromatic amino-acid decarboxylase Inhibitor1 item
- L-Phenylalanine hydroxylase Activator1 item
- L-Tyrosine hydroxylase Inhibitor1 item
- LCK proto-oncogene,Src family tyrosine kinase Inhibitor3item
- LPA1 receptor Antagonist1 item
- LYN proto-oncogene,Src family tyrosine kinase Inhibitor3item
- M1 receptor Agonist1 item
- M1 receptor Allosteric modulator1 item
- M1 receptor Antagonist8item
- M2 receptor Agonist1 item
- M2 receptor Allosteric modulator1 item
- M2 receptor Antagonist8item
- M3 receptor Agonist1 item
- M3 receptor Antagonist8item
- M4 receptor Agonist1 item
- M4 receptor Antagonist8item
- M5 receptor Agonist1 item
- M5 receptor Antagonist7item
- MAPK/ERK Pathway1 item
- Maxi Cl⁻ Activator2item
- MCL1 apoptosis regulator,BCL2 family member Antagonist1 item
- mechanistic target of rapamycin kinase Inhibitor1 item
- MEK1 item
- MET proto-oncogene,receptor tyrosine kinase Inhibitor4item
- Metabolic Enzyme/Protease4item
- mGlu5 receptor Allosteric modulator1 item
- Mineralocorticoid receptor Agonist3item
- Mineralocorticoid receptor Antagonist3item
- mitochondrial pyruvate carrier 1 like Inhibitor1 item
- mitochondrial pyruvate carrier 2 Inhibitor1 item
- mitogen-activated protein kinase kinase 1 Allosteric modulator3item
- mitogen-activated protein kinase kinase 1 Inhibitor1 item
- mitogen-activated protein kinase kinase 2 Allosteric modulator2item
- mitogen-activated protein kinase kinase 2 Inhibitor1 item
- mitogen-activated protein kinase kinase 7 Allosteric modulator1 item
- mitogen-activated protein kinase kinase kinase kinase 5 Inhibitor1 item
- MMP7 Inhibitor1 item
- MMP8 Inhibitor1 item
- Monoamine oxidase A Inhibitor1 item
- Monoamine oxidase B Inhibitor3item
- Monocyclic monoterpenes1 item
- MT1 receptor Agonist1 item
- MT2 receptor Agonist1 item
- Na-Cl symporter Inhibitor3item
- Natural polymer1 item
- Navi2.1 Channel blocker1 item
- NET Inhibitor9item
- Neuronal Signaling1 item
- Neurotransmission1 item
- neurotrophic receptor tyrosine kinase 3 Inhibitor1 item
- nicotinic acetylcholine receptor α1 subunit Antagonist1 item
- nicotinic acetylcholine receptor α3 subunit Agonist1 item
- nicotinic acetylcholine receptor α4 subunit Agonist1 item
- Nitrogenous compounds1 item
- NK1 receptor Antagonist1 item
- OATP1B1 Inhibitor1 item
- OATP1B3 Inhibitor2item
- OATP1C1 Inhibitor1 item
- OATP2B1 Inhibitor2item
- Organic anion transporter 1 Inhibitor1 item
- Ornithine decarboxylase Inhibitor1 item
- P2X4 Antagonist1 item
- P2Y12 receptor Antagonist1 item
- PAR1 Antagonist1 item
- PARP1 item
- PDGFR1 item
- peptidylprolyl isomerase A Inhibitor1 item
- peptidylprolyl isomerase D Inhibitor1 item
- Peroxisome proliferator-activated receptor-α Agonist2item
- Peroxisome proliferator-activated receptor-β/δ Agonist1 item
- Peroxisome proliferator-activated receptor-γ Agonist2item
- Peroxisome proliferator-activated receptor-γ Antagonist2item
- Pharmaceutical ingredients1 item
- phosphatidylinositol 4-kinase type 2 alpha Inhibitor1 item
- phosphatidylinositol 4-kinase type 2 beta Inhibitor1 item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha Inhibitor4item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta Inhibitor3item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta Inhibitor5item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma Inhibitor3item
- phosphodiesterase 11A Inhibitor1 item
- phosphodiesterase 3A Inhibitor5item
- phosphodiesterase 3B Inhibitor2item
- phosphodiesterase 4A Inhibitor2item
- phosphodiesterase 4B Inhibitor2item
- phosphodiesterase 4C Inhibitor2item
- phosphodiesterase 4D Inhibitor1 item
- phosphodiesterase 5A Inhibitor4item
- phosphodiesterase 6C Inhibitor1 item
- phosphodiesterase 7B Inhibitor1 item
- phosphodiesterase 8A Inhibitor1 item
- phosphodiesterase 8B Inhibitor1 item
- Plasma membrane monoamine transporter Inhibitor3item
- plasminogen Inhibitor1 item
- platelet derived growth factor receptor alpha Inhibitor1 item
- platelet derived growth factor receptor beta Inhibitor4item
- polo like kinase 4 Inhibitor1 item
- poly(ADP-ribose) polymerase 1 Inhibitor4item
- poly(ADP-ribose) polymerase 2 Inhibitor3item
- polypeptide1 item
- Pregnane X receptor Agonist1 item
- Progesterone receptor Agonist3item
- proteasome 20S subunit beta 5 Inhibitor1 item
- protein kinase N1 Inhibitor1 item
- Protein Tyrosine Kinase/RTK2item
- Proton-coupled Amino acid Transporter 1 Inhibitor1 item
- Raf-1 proto-oncogene,serine/threonine kinase Inhibitor2item
- RAR-related orphan receptor-β Agonist1 item
- RAR-related orphan receptor-β Antagonist1 item
- receptor interacting serine/threonine kinase 1 Inhibitor1 item
- receptor interacting serine/threonine kinase 2 Inhibitor1 item
- receptor interacting serine/threonine kinase 3 Inhibitor1 item
- Reducing Agents2item
- Regenerative medicine research reagents1 item
- renin Inhibitor1 item
- ret proto-oncogene Inhibitor6item
- Retinoic acid receptor-α Agonist3item
- Retinoic acid receptor-β Agonist3item
- Retinoic acid receptor-γ Agonist3item
- Retinoid X receptor-α Agonist1 item
- Retinoid X receptor-β Agonist1 item
- Retinoid X receptor-γ Agonist1 item
- Rho associated coiled-coil containing protein kinase 1 Inhibitor2item
- Rho associated coiled-coil containing protein kinase 2 Inhibitor2item
- ribonucleotide reductase catalytic subunit M1 Inhibitor2item
- ribonucleotide reductase regulatory subunit M2 Inhibitor2item
- S1P1 receptor Agonist4item
- S1P2 receptor Agonist1 item
- S1P3 receptor Agonist3item
- S1P4 receptor Agonist3item
- S1P5 receptor Agonist4item
- salt inducible kinase 1 Inhibitor2item
- salt inducible kinase 2 Inhibitor2item
- serine/threonine kinase 10 Inhibitor1 item
- serine/threonine kinase 24 Inhibitor1 item
- serine/threonine kinase 4 Inhibitor1 item
- serpin family C member 1 Activator3item
- SERT Inhibitor12item
- Seven membered ring compound2item
- sigma non-opioid intracellular receptor 11 item
- SIK family kinase 3 Inhibitor2item
- SMCT1 Inhibitor1 item
- SMO Antagonist3item
- Sodium/bile acid and sulphated solute cotransporter 1 Inhibitor2item
- Sodium/glucose cotransporter 1 Inhibitor8item
- Sodium/glucose cotransporter 2 Inhibitor8item
- sodium/potassium-transporting ATPase subunit α-1 Inhibitor1 item
- Spectroscopic reagent1 item
- squalene synthase Inhibitor1 item
- SRC proto-oncogene,non-receptor tyrosine kinase Inhibitor4item
- SST2 receptor Agonist1 item
- SST3 receptor Agonist1 item
- SST5 receptor Agonist1 item
- Stem cell biology1 item
- Stem Cell/Wnt1 item
- TAS2R16 Antagonist1 item
- TAS2R31 Agonist1 item
- TAS2R38 Agonist1 item
- TAS2R38 Antagonist1 item
- TAS2R4 Agonist1 item
- TAS2R46 Agonist1 item
- TAS2R9 Agonist1 item
- tec protein tyrosine kinase Inhibitor2item
- Terpenoids1 item
- Testicular receptor 4 Agonist1 item
- testis specific serine kinase 1B Inhibitor1 item
- Thrombopoietin receptor Agonist2item
- thymidylate synthetase Inhibitor1 item
- Thyroid hormone receptor-α Agonist2item
- Thyroid hormone receptor-β Agonist2item
- thyroid peroxidase Inhibitor1 item
- TLR4 Agonist1 item
- TLR7 Antagonist1 item
- TLR9 Antagonist1 item
- TLX Agonist1 item
- TNNI3 interacting kinase Inhibitor1 item
- TP receptor Agonist1 item
- TPC1 Channel blocker1 item
- TPC2 Channel blocker1 item
- TRH1 receptor Agonist1 item
- TRH2 receptor Agonist1 item
- TRPC5 Activator1 item
- TRPC5 Channel blocker2item
- TRPM3 Channel blocker4item
- TRPM4 Channel blocker2item
- TRPM7 Channel blocker1 item
- TRPM8 Activator1 item
- TRPV1 Activator1 item
- TRPV2 Activator1 item
- TRPV4 Activator1 item
- tubulin beta class I Inhibitor5item
- TXK tyrosine kinase Inhibitor3item
- tyrosine kinase 2 Allosteric modulator1 item
- tyrosine kinase 2 Inhibitor6item
- tyrosine kinase non receptor 2 Inhibitor1 item
- UDP-glucose ceramide glucosyltransferase Inhibitor1 item
- V1A receptor Antagonist1 item
- V2 receptor Antagonist1 item
- VEGFR1 item
- Vesicular inhibitory amino acid transporter Inhibitor1 item
- Vesicular monoamine transporter 2 Inhibitor1 item
- Vitamin D receptor Agonist3item
- Vitamin D Related/Nuclear Receptor1 item
- vitamin K epoxide reductase complex subunit 1 Inhibitor3item
- VRAC Activator1 item
- VRAC Channel blocker1 item
- YES proto-oncogene 1,Src family tyrosine kinase Inhibitor1 item
- α1A-adrenoceptor Agonist2item
- α1A-adrenoceptor Antagonist7item
- α1B-adrenoceptor Agonist2item
- α1B-adrenoceptor Antagonist6item
- α1D-adrenoceptor Agonist2item
- α1D-adrenoceptor Antagonist7item
- α2A-adrenoceptor Agonist5item
- α2A-adrenoceptor Antagonist7item
- α2B-adrenoceptor Agonist5item
- α2B-adrenoceptor Antagonist6item
- α2C-adrenoceptor Agonist5item
- α2C-adrenoceptor Antagonist6item
- β1-adrenoceptor Agonist7item
- β1-adrenoceptor Antagonist9item
- β2-adrenoceptor Agonist14item
- β2-adrenoceptor Antagonist7item
- β3-adrenoceptor Agonist4item
- β3-adrenoceptor Antagonist2item
- γ-Glutamyl carboxylase Inhibitor1 item
- δ receptor Antagonist3item
- κ receptor Antagonist3item
- μ receptor Antagonist3item
- ACTIVATOR16item
- AGONIST107item
- ALLOSTERIC MODULATOR7item
- ANTAGONIST120item
- BLOCKER3item
- CHANNEL BLOCKER22item
- GATING INHIBITOR5item
- INHIBITOR215item
- INVERSE AGONIST1 item
- MODULATOR3item
- NEGATIVE ALLOSTERIC MODULATOR2item
- OPENER1 item
- PARTIAL AGONIST3item
- POSITIVE MODULATOR1 item